SCHEMBL5181306

SCHEMBL5181306

O=C(CC(O)CNC(=O)c1ccc(C#Cc2cccc([N+](=O)[O-])c2)cc1)NO

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FFAR1 O14842 1/20 0.47
ATM Q13315 1/20 0.43
ALDH1A1 P00352 5/20 0.43
MAPT P10636 4/20 0.43
HSP90AA1 P07900 2/20 0.43
HTT P42858 2/20 0.43
NPSR1 Q6W5P4 2/20 0.43
S1PR2 O95136 1/20 0.43
OPRK1 P41145 1/20 0.43
HDAC1 Q13547 2/20 0.41
HDAC3 O15379 1/20 0.41
HDAC4 P56524 1/20 0.41
HDAC7 Q8WUI4 1/20 0.41
HDAC2 Q92769 1/20 0.41
HDAC10 Q969S8 1/20 0.41
HDAC11 Q96DB2 1/20 0.41
HDAC8 Q9BY41 1/20 0.41
HDAC6 Q9UBN7 1/20 0.41
HDAC9 Q9UKV0 1/20 0.41
HDAC5 Q9UQL6 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5184545 0.83 GRM5 (0.47) RAB9A
SCHEMBL1105523 0.74 S1PR2 (0.46) FFAR1ALDH1A1MAPTHSP90AA1HTT
SCHEMBL404588 0.74 S1PR2 (0.46) FFAR1ALDH1A1MAPTHSP90AA1HTT
SCHEMBL404589 0.74 S1PR2 (0.46) FFAR1ALDH1A1MAPTHSP90AA1HTT
SCHEMBL404504 0.71 FFAR1 (0.44) FFAR1ALDH1A1MAPTHSP90AA1HTT
SCHEMBL399936 0.71 FFAR1 (0.44) FFAR1ALDH1A1MAPTHSP90AA1HTT
SCHEMBL440373 0.71 HTT (0.45) ALDH1A1MAPTHSP90AA1HTTNPSR1
SCHEMBL5184336 0.70 RAB9A (0.51) ALDH1A1HDAC1HDAC3HDAC4HDAC7
SCHEMBL28728423 0.69 TSHR (0.67) FFAR1ALDH1A1MAPTHSP90AA1HTT
SCHEMBL404493 0.68 BCHE (0.38) ALDH1A1S1PR2HDAC1HDAC8HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1618087-A4 ANTIBACTERIAL AGENTS NOVARTIS VACCINES & DIAGNOSTIC (US) 2007-01-31 EP disclosed
EP-1618087-A2 ANTIBACTERIAL AGENTS CHIRON CORPORATION (US) 2006-01-25 EP disclosed
WO-2004062601-A2 ANTIBACTERIAL AGENTS CHIRON CORPORATION (US) 2004-07-29 WO disclosed