SCHEMBL5184333

SCHEMBL5184333

NC(=O)C[C@@H](C(=O)Nc1nc2ccccc2s1)c1ccccc1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CSNK1D P48730 5/20 0.67
NCS1 P62166 1/20 0.64
ACP1 P24666 3/20 0.60
PTPN7 P35236 1/20 0.60
PTPN12 Q05209 1/20 0.60
PTPN13 Q12923 1/20 0.60
SSU72 Q9NP77 1/20 0.60
SCD O00767 1/20 0.56
SMN1; SMN2 Q16637 3/20 0.53
NPC1 O15118 3/20 0.53
RAB9A P51151 3/20 0.53
MEN1 O00255 2/20 0.53
KMT2A Q03164 2/20 0.53
NFKB1 P19838 2/20 0.53
NFKB2 Q00653 2/20 0.53
RELA Q04206 2/20 0.53
POLB P06746 1/20 0.53
GAA P10253 2/20 0.52
MAPT P10636 2/20 0.52
ALDH1A1 P00352 2/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17287819 1.00 CSNK1D (0.67) CSNK1DNCS1ACP1PTPN7PTPN12
SCHEMBL17287822 0.83 CSNK1D (0.75) CSNK1DNCS1ACP1PTPN7PTPN12
SCHEMBL4244535 0.82 CSNK1D (0.73) CSNK1DNCS1ACP1PTPN7PTPN12
SCHEMBL13949524 0.80 CSNK1D (1.00) CSNK1DNCS1ACP1PTPN7PTPN12
SCHEMBL7362397 0.79 HPGD (0.51) CSNK1DNCS1SMN1; SMN2NPC1RAB9A
SCHEMBL17287798 0.78 CSNK1D (1.00) CSNK1DNCS1ACP1PTPN7PTPN12
SCHEMBL5183402 0.77 MRE11 (0.55) MEN1KMT2APOLBMAPT
SCHEMBL4945628 0.76 CSNK1D (0.60) CSNK1DNCS1ACP1PTPN7PTPN12
SCHEMBL5184192 0.76 CCNE1 (0.53) SMN1; SMN2MEN1KMT2APOLBMAPT
SCHEMBL31078931 0.75 GAA (0.71) CSNK1DACP1SCDSMN1; SMN2NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1758920-A1 BACTERIAL EFFLUX PUMP INHIBITORS AND METHODS OF TREATING BACTERIAL INFECTIONS MPEX PHARMACEUTICALS, INC. (US) 2007-03-07 EP disclosed
WO-2005113579-A1 BACTERIAL EFFLUX PUMP INHIBITORS AND METHODS OF TREATING BACTERIAL INFECTIONS MPEX PHARMACEUTICALS, INC. (US) 2005-12-01 WO disclosed