SCHEMBL5187367

SCHEMBL5187367

CC(=O)Nc1cccc(-c2ccc([C@@H]3CN(C)C[C@H]3NS(=O)(=O)C(C)C)cc2)c1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
GRIA2 P42262 18/20 1.00
KCNH2 Q12809 12/20 1.00
KDM1A O60341 1/20 0.50
BACE1 P56817 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5187358 1.00 GRIA2 (1.00) GRIA2KCNH2KDM1ABACE1
SCHEMBL5187342 1.00 GRIA2 (1.00) GRIA2KCNH2KDM1ABACE1
SCHEMBL4958828 0.88 GRIA2 (1.00) GRIA2KCNH2
SCHEMBL5456189 0.86 GRIA2 (1.00) GRIA2KCNH2KDM1A
SCHEMBL4956505 0.86 GRIA2 (1.00) GRIA2KCNH2KDM1A
SCHEMBL4607084 0.85 GRIA2 (0.74) GRIA2KCNH2KDM1A
SCHEMBL7250835 0.85 GRIA2 (0.74) GRIA2KCNH2KDM1A
SCHEMBL7250833 0.85 GRIA2 (0.74) GRIA2KCNH2KDM1A
SCHEMBL5450587 0.82 GRIA2 (0.72) GRIA2KCNH2
SCHEMBL4955429 0.82 GRIA2 (0.72) GRIA2KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20070270471-A1 Compounds Which Potentiate Glutamate Receptor and Uses Thereof in Medicine GLAXO GROUP LIMITED (GB) 2007-11-22 US claimed
US-20070270471-A1 Compounds Which Potentiate Glutamate Receptor and Uses Thereof in Medicine GLAXO GROUP LIMITED (GB) 2007-11-22 US disclosed
EP-1786769-A1 COMPOUNDS WHICH POTENTIATE GLUTAMATE RECEPTOR AND USES THEREOF IN MEDICINE GLAXO GROUP LIMITED (GB) 2007-05-23 EP disclosed
WO-2006015827-A1 COMPOUNDS WHICH POTENTIATE GLUTAMATE RECEPTOR AND USES THEREOF IN MEDICINE GLAXO GROUP LIMITED (GB) 2006-02-16 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070270471-A1 Compounds Which Potentiate Glutamate Receptor and Uses Thereof in Medicine GRM3, GLRA3, GLRA1 GRIA2 34/4885KCNH2 562/4885KDM1A 3089/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.