SCHEMBL5190571

SCHEMBL5190571

O=C(CC1CNCCN1)NC(=O)Nc1ccccc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
JAK3 P52333 2/20 0.47
SMN1; SMN2 Q16637 2/20 0.41
EPHX2 P34913 2/20 0.41
EPHX1 P07099 2/20 0.41
TP53 P04637 1/20 0.41
TSHR P16473 1/20 0.41
CDK9 P50750 1/20 0.41
CLK4 Q9HAZ1 1/20 0.41
MEN1 O00255 1/20 0.41
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
KMT2A Q03164 1/20 0.41
LTA4H P09960 1/20 0.40
ALDH1A1 P00352 1/20 0.40
MAP2K1 Q02750 1/20 0.39
GAA P10253 2/20 0.39
TAAR1 Q96RJ0 1/20 0.39
PKM P14618 1/20 0.39
FPR1 P21462 2/20 0.38
FPR2 P25090 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5193257 0.80 PPARG (0.39) EPHX2LTA4H
SCHEMBL21162505 0.76 MC4R (0.52) JAK3SMN1; SMN2MEN1NPC1RAB9A
SCHEMBL5231090 0.73 GAA (0.48) SMN1; SMN2EPHX2TSHRMEN1RAB9A
SCHEMBL27456628 0.73 KMT2A (0.48) SMN1; SMN2TP53MEN1NPC1RAB9A
SCHEMBL28402347 0.73 NPC1 (0.48) SMN1; SMN2TP53TSHRMEN1NPC1
SCHEMBL3829656 0.72 KMT2A (0.46) EPHX1MEN1KMT2AALDH1A1GAA
SCHEMBL5195330 0.71 CHRNB2 (0.37) EPHX2EPHX1MEN1KMT2AALDH1A1
SCHEMBL5189969 0.70 EPHX1 (0.47) SMN1; SMN2EPHX2EPHX1NPC1RAB9A
SCHEMBL5193666 0.70 HTT (0.46) SMN1; SMN2TSHRMEN1NPC1RAB9A
SCHEMBL5190160 0.70

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0968206-B8 N-HETEROCYCLIC DERIVATIVES AS NOS INHIBITORS BERLEX INC (US) 2007-01-24 EP disclosed
EP-0968206-A1 N-HETEROCYCLIC DERIVATIVES AS NOS INHIBITORS BERLEX LABORATORIES, INC. (US) 2000-01-05 EP disclosed
WO-1998037079-A1 N-HETEROCYCLIC DERIVATIVES AS NOS INHIBITORS BERLEX LABORATORIES, INC. (US) 1998-08-27 WO disclosed