SCHEMBL5192064

SCHEMBL5192064

Cc1cc(N2CCOC(C(=O)NC(C)c3ccc4c(c3)OCCO4)C2)nc(-n2ccnc2)n1

nearest known ligand 0.51

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
NOS2 P35228 16/20 0.51
NOS1 P29475 1/20 0.43
HTT P42858 2/20 0.43
KDM4E B2RXH2 1/20 0.41
MEN1 O00255 1/20 0.40
USP2 O75604 1/20 0.40
KMT2A Q03164 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5191340 0.96 NOS2 (0.56) NOS2NOS1
SCHEMBL5192349 0.91 NOS2 (0.46) NOS2HTT
SCHEMBL5192204 0.88 NOS2 (0.44) NOS2
SCHEMBL5190216 0.88 NOS2 (0.45) NOS2
SCHEMBL5193161 0.87 NOS2 (0.49) NOS2
SCHEMBL5192066 0.84 NOS2 (0.66) NOS2NOS1
SCHEMBL5190610 0.84 NOS2 (0.65) NOS2NOS1HTT
SCHEMBL5192623 0.83 NOS2 (0.55) NOS2NOS1MEN1USP2KMT2A
SCHEMBL5192225 0.83 NOS2 (0.53) NOS2NOS1
SCHEMBL5191677 0.82 NOS2 (0.62) NOS2NOS1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1754703-A2 N-Heterocyclic derivatives as nos inhibitors Berlex, Inc. (US) 2007-02-21 EP claimed
EP-1754703-A2 N-Heterocyclic derivatives as nos inhibitors Berlex, Inc. (US) 2007-02-21 EP disclosed
EP-0968206-B1 N-HETEROCYCLIC DERIVATIVES AS NOS INHIBITORS BERLEX LAB (US) 2006-11-15 EP disclosed
CN-1100777-C N-heterocyclic derivatives as NOS inhibitor BERLEX LAB (US) 2003-02-05 CN disclosed
CN-1252799-A N-heterocyclic derivatives as NOS inhibitor BERLEX LAB (US) 2000-05-10 CN disclosed