SCHEMBL5195657

SCHEMBL5195657

CCCCC=C(NC(=O)OCc1ccccc1)C(=O)O

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.46
CYP3A4 P08684 1/20 0.46
TSHR P16473 1/20 0.46
MAPK1 P28482 1/20 0.46
TDP1 Q9NUW8 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
CA12 O43570 1/20 0.45
CA1 P00915 1/20 0.45
CA2 P00918 1/20 0.45
CA9 Q16790 1/20 0.45
CTSL P07711 1/20 0.45
CTSS P25774 1/20 0.45
NPC1 O15118 1/20 0.44
RAB9A P51151 1/20 0.44
HTT P42858 1/20 0.44
SMN1; SMN2 Q16637 2/20 0.43
MBOAT4 Q96T53 1/20 0.43
LMNA P02545 1/20 0.43
TGM2 P21980 1/20 0.42
PRTN3 P24158 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5195650 1.00 ALDH1A1 (0.46) ALDH1A1CYP3A4TSHRMAPK1TDP1
SCHEMBL5195644 1.00 ALDH1A1 (0.46) ALDH1A1CYP3A4TSHRMAPK1TDP1
SCHEMBL5412247 0.90 ALDH1A1 (0.44) ALDH1A1CYP3A4TSHRMAPK1TDP1
SCHEMBL5412244 0.90 ALDH1A1 (0.44) ALDH1A1CYP3A4TSHRMAPK1TDP1
SCHEMBL6822887 0.87 CA12 (0.45) ALDH1A1CA12CA1CA2CA9
SCHEMBL6822885 0.87 CA12 (0.45) ALDH1A1CA12CA1CA2CA9
SCHEMBL6822886 0.87 CA12 (0.45) ALDH1A1CA12CA1CA2CA9
SCHEMBL2855446 0.85 CA12 (0.48) ALDH1A1CA12CA1CA2CA9
SCHEMBL2855442 0.85 CA12 (0.48) ALDH1A1CA12CA1CA2CA9
SCHEMBL4245008 0.82 CA12 (0.50) ALDH1A1MAPK1TDP1L3MBTL1CA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1812383-A1 GLYCOGEN PHOSPHORYLASE INHIBITOR COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS THEREOF Smithkline Beecham Corporation (US) 2007-08-01 EP disclosed
WO-2006052722-A1 GLYCOGEN PHOSPHORYLASE INHIBITOR COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS THEREOF SMITHKLINE BEECHAM CORPORATION (US) 2006-05-18 WO disclosed