SCHEMBL5197409

SCHEMBL5197409

CC(C)(C)NC(=O)OC1Cc2ccccc2CN1C1CCCc2cc(Oc3ccc(C(N)=O)cn3)ccc21

nearest known ligand 0.48

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 19/20 0.48
OPRD1 P41143 18/20 0.48
OPRK1 P41145 15/20 0.48
HRH3 Q9Y5N1 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL387332 0.89 OPRM1 (0.49) OPRM1OPRD1OPRK1HRH3
SCHEMBL388331 0.78 HRH3 (0.64) OPRM1OPRD1OPRK1HRH3
SCHEMBL388149 0.73 HRH3 (0.64) OPRM1OPRD1OPRK1HRH3
SCHEMBL14378986 0.73 HRH3 (0.59) OPRM1OPRD1OPRK1HRH3
SCHEMBL385447 0.73 HRH3 (0.56) OPRM1OPRD1OPRK1HRH3
SCHEMBL389441 0.72 HRH3 (0.59) OPRM1OPRD1OPRK1HRH3
SCHEMBL387361 0.72 HRH3 (0.60) OPRM1OPRD1OPRK1HRH3
SCHEMBL385666 0.71 HRH3 (0.59) OPRM1OPRD1OPRK1HRH3
SCHEMBL385483 0.69 HRH3 (0.57) OPRM1OPRD1OPRK1HRH3
SCHEMBL10175569 0.69 HRH3 (0.57) OPRM1OPRD1OPRK1HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1613597-B1 6-SUBSTITUTED NICOTINAMIDE DERIVATIVES AS OPIOID RECEPTOR ANTAGONISTS LILLY CO ELI (US) 2007-11-07 EP claimed