SCHEMBL5198581

SCHEMBL5198581

CCCCN1C(=O)C(NCc2ccc3c(c2)OCO3)=C(c2ccccc2)S1(=O)=O.COCCN1C(=O)C(NC2Cc3ccccc3C2)=C(c2ccccc2)S1(=O)=O.O=C1C(NCCCCc2ccccc2)=C(c2ccccc2)S(=O)(=O)N1Cc1ccncc1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.35
TSHR P16473 2/20 0.35
GAA P10253 2/20 0.35
HPGD P15428 1/20 0.35
LMNA P02545 2/20 0.34
L3MBTL1 Q9Y468 2/20 0.34
ACHE P22303 1/20 0.33
BACE1 P56817 1/20 0.33
FLT1 P17948 2/20 0.33
KDR P35968 2/20 0.33
TDP1 Q9NUW8 1/20 0.33
PSEN1 P49768 1/20 0.33
PSEN2 P49810 1/20 0.33
APH1B Q8WW43 1/20 0.33
NCSTN Q92542 1/20 0.33
APH1A Q96BI3 1/20 0.33
PSENEN Q9NZ42 1/20 0.33
ALDH1A1 P00352 6/20 0.32
HTT P42858 1/20 0.32
HIF1A Q16665 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1999415 0.77 HPGD (0.48) SMN1; SMN2TSHRGAAHPGDL3MBTL1
SCHEMBL2001526 0.76 SMN1; SMN2 (0.52) SMN1; SMN2TSHRGAAHPGDLMNA
SCHEMBL2001043 0.72 ASAH1 (0.41) SMN1; SMN2HIF1AKDM4E
SCHEMBL1997463 0.71 HPGD (0.36) SMN1; SMN2GAAHPGDALDH1A1KDM4E
SCHEMBL5200606 0.70 MEN1 (0.38) SMN1; SMN2TSHRGAAHPGDLMNA
SCHEMBL2000476 0.68 CA12 (0.40) ACHEMAPK1
SCHEMBL5185942 0.68 ACHE (0.43) GAAHPGDL3MBTL1ACHEALDH1A1
SCHEMBL2000223 0.67 CA12 (0.44) SMN1; SMN2L3MBTL1ALDH1A1KDM4E
SCHEMBL1998233 0.66 CA12 (0.45) SMN1; SMN2GAAACHEALDH1A1KMT2A
SCHEMBL19127183 0.66 CA12 (0.40) SMN1; SMN2TSHRGAAHPGDLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1838687-A1 NON-ANILINIC DERIVATIVES OF ISOTHIAZOL-3(2H)-ONE 1,1-DIOXIDES AS LIVER X RECEPTOR MODULATORS AstraZeneca AB (SE) 2007-10-03 EP disclosed
WO-2006073366-A1 NON-ANILINIC DERIVATIVES OF ISOTHIAZOL-3(2H)-ONE 1,1-DIOXIDES AS LIVER X RECEPTOR MODULATORS ASTRAZENECA AB (SE) 2006-07-13 WO disclosed