SCHEMBL5199712

SCHEMBL5199712

Cc1cc(C#Cc2ccc(-c3ccc(Cl)cc3)cn2)ccc1OCC[C]1CCCC1

nearest known ligand 0.64

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 19/20 0.64
CHRM1 P11229 4/20 0.64
HTR2A P28223 3/20 0.49
CYP2D6 P10635 1/20 0.49
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2C19 P33261 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5230359 0.99 MCHR1 (0.63) MCHR1CHRM1HTR2ACYP2D6CYP1A2
SCHEMBL2319440 0.85 MCHR1 (0.68) MCHR1CHRM1HTR2ACYP2D6CYP1A2
SCHEMBL2321296 0.83 MCHR1 (0.82) MCHR1CHRM1HTR2ACYP2D6
SCHEMBL5199790 0.83 MCHR1 (0.66) MCHR1CHRM1HTR2ACYP2D6
SCHEMBL4491965 0.83 MCHR1 (0.63) MCHR1CHRM1HTR2ACYP2D6CYP1A2
SCHEMBL4489001 0.83 MCHR1 (0.63) MCHR1CHRM1HTR2ACYP2D6CYP1A2
SCHEMBL2328524 0.82 MCHR1 (0.80) MCHR1CHRM1HTR2ACYP2D6
SCHEMBL2322440 0.82 MCHR1 (0.80) MCHR1CHRM1HTR2ACYP2D6
SCHEMBL4471247 0.82 MCHR1 (0.62) MCHR1CHRM1HTR2ACYP2D6CYP1A2
SCHEMBL2323226 0.82 MCHR1 (0.69) MCHR1CHRM1HTR2ACYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1737823-A2 NOVEL ALKYNE COMPOUNDS WITH AN MCH-ANTAGONISTIC ACTION AND MEDICAMENTS COMPRISING SAID COMPOUNDS Boehringer Ingelheim International GmbH (DE) 2007-01-03 EP disclosed
WO-2005103002-A2 NOVEL ALKYNE COMPOUNDS WITH AN MCH-ANTAGONISTIC ACTION AND MEDICAMENTS COMPRISING SAID COMPOUNDS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2005-11-03 WO disclosed