SCHEMBL5199790

SCHEMBL5199790

Clc1ccc(-c2ccc(C#Cc3ccc(OCC[C]4CCCCC4)cc3)nc2)cc1

nearest known ligand 0.66

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 20/20 0.66
CHRM1 P11229 3/20 0.66
HTR2A P28223 3/20 0.66
CYP2D6 P10635 1/20 0.66

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5230359 0.84 MCHR1 (0.63) MCHR1CHRM1HTR2ACYP2D6
SCHEMBL5199712 0.83 MCHR1 (0.64) MCHR1CHRM1HTR2ACYP2D6
SCHEMBL2323590 0.82 MCHR1 (0.69) MCHR1CHRM1HTR2ACYP2D6
SCHEMBL2319087 0.81 MCHR1 (0.98) MCHR1CHRM1HTR2ACYP2D6
SCHEMBL2321590 0.80 MCHR1 (0.96) MCHR1CHRM1HTR2ACYP2D6
SCHEMBL2326502 0.80 MCHR1 (1.00) MCHR1CHRM1HTR2ACYP2D6
SCHEMBL4474659 0.78 MCHR1 (0.58) MCHR1CHRM1HTR2ACYP2D6
SCHEMBL5198730 0.78 MCHR1 (0.63) MCHR1CHRM1HTR2ACYP2D6
SCHEMBL4521439 0.78 MCHR1 (0.72) MCHR1CHRM1HTR2ACYP2D6
SCHEMBL4475403 0.77 MCHR1 (0.57) MCHR1CHRM1HTR2ACYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1737823-A2 NOVEL ALKYNE COMPOUNDS WITH AN MCH-ANTAGONISTIC ACTION AND MEDICAMENTS COMPRISING SAID COMPOUNDS Boehringer Ingelheim International GmbH (DE) 2007-01-03 EP claimed
WO-2005103002-A2 NOVEL ALKYNE COMPOUNDS WITH AN MCH-ANTAGONISTIC ACTION AND MEDICAMENTS COMPRISING SAID COMPOUNDS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2005-11-03 WO claimed