SCHEMBL5200710

SCHEMBL5200710

O=Cc1cc(C[C@@H]2CNCCO2)ccc1O

nearest known ligand 0.48

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CDK1 P06493 1/20 0.44
ERN1 O75460 7/20 0.36
NT5E P21589 1/20 0.35
DRD2 P14416 1/20 0.35
DRD3 P35462 1/20 0.35
SLC6A2 P23975 3/20 0.34
SLC6A4 P31645 3/20 0.34
SLC6A3 Q01959 3/20 0.34
ADRB2 P07550 1/20 0.34
HTR1A P08908 1/20 0.34
HTR2A P28223 1/20 0.34
ADRA1A P35348 1/20 0.34
HTR2B P41595 1/20 0.34
ADRA2C P18825 1/20 0.34
ESR2 Q92731 1/20 0.34
CYP19A1 P11511 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5200714 1.00 CDK1 (0.44) CDK1ERN1NT5EDRD2DRD3
SCHEMBL27695212 0.80 DRD2 (0.40) DRD2DRD3SLC6A2SLC6A4SLC6A3
SCHEMBL5184704 0.80 DRD2 (0.40) DRD2DRD3SLC6A2SLC6A4SLC6A3
SCHEMBL6834244 0.78 SLC6A2 (0.39) SLC6A2SLC6A4SLC6A3ADRB2HTR1A
SCHEMBL1929978 0.77 DRD2 (0.40) DRD2DRD3SLC6A2SLC6A4SLC6A3
SCHEMBL1551829 0.76 DRD2 (0.42) DRD2DRD3SLC6A2SLC6A4SLC6A3
SCHEMBL27828941 0.76 DRD2 (0.42) DRD2DRD3SLC6A2SLC6A4SLC6A3
SCHEMBL21249083 0.75 DRD2 (0.56) DRD2DRD3SLC6A3HTR1AESR2
SCHEMBL27537852 0.74 DRD2 (0.55) DRD2DRD3SLC6A2SLC6A4SLC6A3
SCHEMBL16759290 0.74 SLC6A2 (0.50) SLC6A2SLC6A4SLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1844026-A2 MORPHOLINES AS 5HT2C AGONISTS F.HOFFMANN-LA ROCHE AG (CH) 2007-10-17 EP disclosed
WO-2006077025-A2 MORPHOLINES AS 5HT2C AGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2006-07-27 WO disclosed