SCHEMBL5200730

SCHEMBL5200730

CCCOc1cccc(C(=O)Cl)c1

nearest known ligand 0.73

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.73
NR1H4 Q96RI1 1/20 0.57
SMPD1 P17405 3/20 0.55
SMN1; SMN2 Q16637 3/20 0.53
NPC1 O15118 3/20 0.53
RAB9A P51151 3/20 0.53
KAT6A Q92794 1/20 0.53
ALDH1A1 P00352 1/20 0.53
LMNA P02545 1/20 0.53
TSHR P16473 1/20 0.53
MAPK1 P28482 1/20 0.53
MAPT P10636 2/20 0.52
PLA2G4B P0C869 1/20 0.51
ADRB2 P07550 1/20 0.51
ADRB1 P08588 1/20 0.51
ADRB3 P13945 1/20 0.51
THRA P10827 1/20 0.50
THRB P10828 1/20 0.50
MEN1 O00255 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5202638 0.92 KMT2A (0.62) KMT2ANR1H4SMPD1KAT6ALMNA
SCHEMBL8465014 0.90 SMPD1 (0.68) KMT2ANR1H4SMPD1TSHRPLA2G4B
SCHEMBL9906433 0.89 SMPD1 (0.70) KMT2ANR1H4SMPD1TSHRPLA2G4B
SCHEMBL9305977 0.89 SMPD1 (0.70) KMT2ANR1H4SMPD1TSHRPLA2G4B
SCHEMBL15779400 0.89 SMPD1 (0.70) KMT2ANR1H4SMPD1TSHRPLA2G4B
SCHEMBL5204104 0.89 SMPD1 (0.70) KMT2ANR1H4SMPD1TSHRPLA2G4B
SCHEMBL11337002 0.89 SMPD1 (0.70) KMT2ANR1H4SMPD1TSHRPLA2G4B
SCHEMBL1331352 0.89 SMPD1 (0.70) KMT2ANR1H4SMPD1TSHRPLA2G4B
SCHEMBL11422303 0.86 PRSS1 (0.60) KMT2ASMPD1PLA2G4BTHRATHRB
SCHEMBL27913517 0.86 KMT2A (0.78) KMT2ANR1H4SMPD1SMN1; SMN2NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117304205-A Benzimidazole ternary fused ring compound, pharmaceutically acceptable salt thereof and application thereof 中国科学院广州生物医药与健康研究院 2023-12-29 CN disclosed
EP-1087946-B1 ARYL ALKANOYLPYRIDAZINES MERCK PATENT GMBH (DE) 2007-01-10 EP disclosed
CN-1168720-C Aryl alkanoylpyridazines Ĭ��ר���ɷ����޹�˾ 2004-09-29 CN disclosed
US-6417188-B1 ENZYME INHIBITORS OF PHOSPHODIESTERASE MERCK PATENT GESELLSCHAFT MIT BESCHRAENKTER HAFTUNG (DE) 2002-07-09 US disclosed
CN-1305465-A Aryl alkanoylpyridazines MERCK PATENT GMBH (DE) 2001-07-25 CN disclosed
EP-1087946-A1 ARYL ALKANOYLPYRIDAZINES MERCK PATENT GmbH (DE) 2001-04-04 EP disclosed
WO-1999065880-A1 ARYL ALKANOYLPYRIDAZINES MERCK PATENT GMBH (DE) 1999-12-23 WO disclosed
US-4001426-A HAVING CORONARY VASODILATOR ACTIVITY SMITHKLINE CORPORATION (US) 1977-01-04 US disclosed