SCHEMBL5200837

SCHEMBL5200837

N#CCCc1cc(Cl)ccc1-c1ccccc1.OCCc1ccccc1-c1ccc(Cl)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FFAR4 Q5NUL3 3/20 0.39
FFAR1 O14842 2/20 0.39
CYP2C19 P33261 1/20 0.36
ADORA2A P29274 1/20 0.36
ADORA1 P30542 1/20 0.36
TSHR P16473 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
ADRA2C P18825 1/20 0.36
PTGDR2 Q9Y5Y4 1/20 0.35
MEN1 O00255 1/20 0.35
POLB P06746 1/20 0.35
KMT2A Q03164 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
HSD17B3 P37058 1/20 0.35
SQOR Q9Y6N5 1/20 0.35
CNR1 P21554 4/20 0.35
PTGER1 P34995 1/20 0.35
PTGER4 P35408 1/20 0.35
PTGER3 P43115 1/20 0.35
PTGER2 P43116 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3732787 0.88 FFAR1 (0.43) FFAR4FFAR1ADORA2AADORA1TSHR
SCHEMBL3746249 0.82 FFAR1 (0.50) FFAR4FFAR1TSHRNPSR1PTGDR2
SCHEMBL3746992 0.79 CYP2C19 (0.50) FFAR4FFAR1CYP2C19NPSR1PTGDR2
SCHEMBL9284366 0.79 DPP4 (0.50) FFAR4FFAR1ADRA2CMEN1KMT2A
SCHEMBL9184322 0.72 MEN1 (0.43) FFAR4FFAR1TSHRMEN1KMT2A
SCHEMBL27840283 0.72 DPP4 (0.58) FFAR4FFAR1KMT2ATDP1PTGER1
SCHEMBL429540 0.72 DPP4 (0.58) FFAR4FFAR1KMT2ATDP1PTGER1
SCHEMBL7791575 0.72 PTGER1 (0.40) FFAR4FFAR1TSHRADRA2CMEN1
SCHEMBL27658164 0.71 DPP4 (0.48) ADRA2CKMT2APTGER1PTGER4PTGER3
SCHEMBL554701 0.71 CYP2C19 (0.45) FFAR4FFAR1CYP2C19ADORA2AADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1817031-A1 NOVEL SPECIFIC CASPASE-10 INHIBITORS Merck Patent GmbH (DE) 2007-08-15 EP claimed
WO-2006058592-A1 NOVEL SPECIFIC CASPASE-10 INHIBITORS MERCK PATENT GMBH (DE) 2006-06-08 WO claimed