SCHEMBL5201601

SCHEMBL5201601

CS(=O)(=O)Nc1cccc(OCC2=NCCN2)c1

nearest known ligand 0.56

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
NISCH Q9Y2I1 10/20 0.56
MAOA P21397 2/20 0.56
MAOB P27338 2/20 0.56
ADRA1A P35348 5/20 0.53
DRD2 P14416 1/20 0.46
DRD4 P21917 1/20 0.46
DRD3 P35462 1/20 0.46
HTR1A P08908 2/20 0.45
ADRA2A P08913 2/20 0.45
ADRA2B P18089 2/20 0.45
ADRA2C P18825 2/20 0.45
ADRA1D P25100 2/20 0.43
ADRA1B P35368 2/20 0.43
HTR1B P28222 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL5202978 0.99 NISCH (0.54) NISCHMAOAMAOBADRA1ADRD2
Hydrochloric Acid SCHEMBL5203127 0.98 NISCH (0.53) NISCHMAOAMAOBADRA1ADRD2
Hydrochloric Acid SCHEMBL8547827 0.88 NISCH (0.53) NISCHMAOAMAOBADRA1AHTR1A
SCHEMBL5203397 0.88 NISCH (0.56) NISCHMAOAMAOBADRA1AHTR1A
Hydrochloric Acid SCHEMBL5201622 0.87 NISCH (0.55) NISCHMAOAMAOBADRA1AHTR1A
SCHEMBL5233626 0.85 NISCH (0.59) NISCHMAOAMAOBADRA1AHTR1A
Hydrochloric Acid SCHEMBL5204122 0.84 NISCH (0.57) NISCHMAOAMAOBADRA1AHTR1A
SCHEMBL5202794 0.83 ADRA1A (0.53) NISCHMAOAMAOBADRA1AHTR1A
SCHEMBL5206670 0.82 ADRA1A (0.49) NISCHMAOAMAOBADRA1AHTR1A
SCHEMBL5203438 0.82 ADRA1A (0.54) NISCHMAOAMAOBADRA1AHTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0887346-B1 N-Phenyl-alkylsulfonamide derivatives, their preparation and their use as alpha1A/1L adrenoceptor agonists HOFFMANN LA ROCHE (CH) 2007-12-12 EP claimed
EP-0887346-A2 Phenyl-and aminophenyl-alkylsulfonamide and urea derivatives, their preparation and their use as alpha1A/1L adrenoceptor agonists F. HOFFMANN-LA ROCHE AG (CH) 1998-12-30 EP claimed
EP-0887346-B1 N-Phenyl-alkylsulfonamide derivatives, their preparation and their use as alpha1A/1L adrenoceptor agonists HOFFMANN LA ROCHE (CH) 2007-12-12 EP disclosed
EP-0887346-B1 N-Phenyl-alkylsulfonamide derivatives, their preparation and their use as alpha1A/1L adrenoceptor agonists HOFFMANN LA ROCHE (CH) 2007-12-12 EP disclosed
EP-0887346-A2 Phenyl-and aminophenyl-alkylsulfonamide and urea derivatives, their preparation and their use as alpha1A/1L adrenoceptor agonists F. HOFFMANN-LA ROCHE AG (CH) 1998-12-30 EP disclosed