SCHEMBL5201643

SCHEMBL5201643

Cc1ccccc1-c1[c]ccc(N)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PLA2G7 Q13093 1/20 0.43
NPC1 O15118 4/20 0.40
RAB9A P51151 4/20 0.40
SMN1; SMN2 Q16637 4/20 0.40
TP53 P04637 2/20 0.40
TSHR P16473 2/20 0.40
KDM4E B2RXH2 1/20 0.40
MAPT P10636 1/20 0.40
HSD17B10 Q99714 1/20 0.40
CYP3A4 P08684 2/20 0.39
TDP1 Q9NUW8 2/20 0.39
CASP1 P29466 1/20 0.38
CTSD P07339 1/20 0.35
BACE1 P56817 1/20 0.35
ALDH1A1 P00352 3/20 0.34
DHFR P00374 1/20 0.34
ADORA2A P29274 1/20 0.33
LCK P06239 1/20 0.33
KDR P35968 1/20 0.33
JAK3 P52333 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3912578 0.81 NPC1 (0.35) NPC1RAB9ASMN1; SMN2TP53TSHR
SCHEMBL9523594 0.78 NPC1 (0.40) PLA2G7NPC1RAB9ASMN1; SMN2TSHR
SCHEMBL9004856 0.78 ESR2 (0.39) NPC1RAB9ASMN1; SMN2TP53TSHR
SCHEMBL8129685 0.78 PDE10A (0.36) NPC1RAB9ASMN1; SMN2TSHRKDM4E
SCHEMBL7467097 0.76 NPC1 (0.39) NPC1RAB9ASMN1; SMN2TSHRKDM4E
SCHEMBL714181 0.76 TSHR (0.41) NPC1RAB9ASMN1; SMN2TSHRCYP3A4
SCHEMBL8125196 0.75 CYP1A2 (0.40) NPC1RAB9ASMN1; SMN2TSHRKDM4E
SCHEMBL9599597 0.75 NPC1 (0.40) NPC1RAB9ASMN1; SMN2TSHRMAPT
SCHEMBL16862586 0.75 DPP4 (0.44) NPC1RAB9ASMN1; SMN2TP53TSHR
SCHEMBL10888098 0.75 CYP1A2 (0.38) NPC1RAB9ASMN1; SMN2TSHRMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1560809-B1 CYCLOHEXYLUREA DERIVATIVES GRUENENTHAL GMBH (DE) 2007-08-22 EP claimed
EP-1560809-A1 CYCLOHEXYLUREA DERIVATIVES Grünenthal GmbH (DE) 2005-08-10 EP claimed
WO-2004043909-A1 CYCLOHEXYLUREA DERIVATIVES Grünenthal GmbH (DE) 2004-05-27 WO claimed
EP-1560809-B1 CYCLOHEXYLUREA DERIVATIVES GRUENENTHAL GMBH (DE) 2007-08-22 EP disclosed
EP-1560809-A1 CYCLOHEXYLUREA DERIVATIVES Grünenthal GmbH (DE) 2005-08-10 EP disclosed
WO-2004043909-A1 CYCLOHEXYLUREA DERIVATIVES Grünenthal GmbH (DE) 2004-05-27 WO disclosed