SCHEMBL8129685

SCHEMBL8129685

Cc1ccccc1-c1[c]ccc(F)c1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE10A Q9Y233 3/20 0.36
PDE2A O00408 2/20 0.36
MAPT P10636 3/20 0.36
POLB P06746 2/20 0.36
MAPK1 P28482 2/20 0.36
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
ALDH1A1 P00352 1/20 0.36
LMNA P02545 1/20 0.36
RECQL P46063 1/20 0.36
ACHE P22303 3/20 0.35
KDM4E B2RXH2 1/20 0.35
ALOX15 P16050 1/20 0.35
ALOX12 P18054 1/20 0.35
HSD17B10 Q99714 1/20 0.35
CYP1A2 P05177 2/20 0.34
CYP3A4 P08684 2/20 0.34
CYP2D6 P10635 2/20 0.34
HPGD P15428 2/20 0.34
CYP2C19 P33261 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8129595 0.86 ACHE (0.35) MAPTPOLBMAPK1MEN1KMT2A
SCHEMBL9650055 0.83 PTGS2 (0.37) PDE10APDE2AACHE
SCHEMBL3912578 0.81 NPC1 (0.35) MAPTMAPK1MEN1KMT2AALDH1A1
SCHEMBL434431 0.81 L3MBTL1 (0.38) ALDH1A1KDM4ECYP1A2HPGDNPC1
SCHEMBL8125196 0.79 CYP1A2 (0.40) MAPTMAPK1MEN1KMT2AALDH1A1
SCHEMBL9138237 0.78 HSD11B1 (0.41) PDE10APDE2APOLBMAPK1MEN1
SCHEMBL9523594 0.78 NPC1 (0.40) PDE10APDE2AMAPTMAPK1MEN1
SCHEMBL5201643 0.78 PLA2G7 (0.43) MAPTPOLBMAPK1MEN1KMT2A
SCHEMBL8077591 0.78 PTGS2 (0.36) MAPTMAPK1ALDH1A1HSD17B10HPGD
SCHEMBL9004856 0.78 ESR2 (0.39) MAPTPOLBMEN1KMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1028945-A1 SUBSTITUTED PYRIDINE COMPOUNDS AS ANTI-INFLAMMATORY AGENTS Amgen Inc. (US) 2000-08-23 EP disclosed
WO-1999024404-A1 SUBSTITUTED PYRIDINE COMPOUNDS AS ANTI-INFLAMMATORY AGENTS AMGEN INC. (US) 1999-05-20 WO disclosed