SCHEMBL5201858

SCHEMBL5201858

O=C(O)Cc1cc([N+](=O)[O-])ccc1-c1ccc(C(F)(F)F)cc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PSEN1 P49768 1/20 0.54
PSEN2 P49810 1/20 0.54
APH1B Q8WW43 1/20 0.54
NCSTN Q92542 1/20 0.54
APH1A Q96BI3 1/20 0.54
PSENEN Q9NZ42 1/20 0.54
CYP1A2 P05177 1/20 0.51
AKR1C3 P42330 2/20 0.46
AKR1C2 P52895 2/20 0.46
RXRA P19793 4/20 0.43
RXRB P28702 4/20 0.43
RXRG P48443 4/20 0.43
RORC P51449 1/20 0.43
PTGDR2 Q9Y5Y4 1/20 0.41
APP P05067 1/20 0.41
ALKBH5 Q6P6C2 1/20 0.41
PHGDH O43175 1/20 0.41
PTGS2 P35354 2/20 0.40
MEN1 O00255 1/20 0.40
LMNA P02545 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3737498 0.83 CYP1A2 (0.55) CYP1A2PTGDR2PTGS2MEN1LMNA
SCHEMBL3736961 0.83 CYP1A2 (0.55) CYP1A2PTGDR2PTGS2MEN1LMNA
SCHEMBL9890672 0.80 PSEN1 (0.61) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL3740107 0.80 CYP1A2 (0.51) CYP1A2APPMEN1LMNAMAPT
SCHEMBL9890676 0.79 PSEN1 (0.59) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL9892653 0.76 PSEN1 (0.56) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL4649430 0.76 APP (0.51) AKR1C3AKR1C2RORCAPPPTGS2
SCHEMBL9892659 0.76 PTGDR2 (0.59) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL27928945 0.75 CYP3A4 (0.46) AKR1C3AKR1C2PTGS2MEN1LMNA
SCHEMBL4937999 0.75 CYP1A2 (0.63) CYP1A2AKR1C3AKR1C2RXRARXRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1817031-A1 NOVEL SPECIFIC CASPASE-10 INHIBITORS Merck Patent GmbH (DE) 2007-08-15 EP disclosed
WO-2006058592-A1 NOVEL SPECIFIC CASPASE-10 INHIBITORS MERCK PATENT GMBH (DE) 2006-06-08 WO disclosed