SCHEMBL5202158

SCHEMBL5202158

N[C@](CC1c2ccccc2Oc2ccccc21)(C(=O)O)C1C[C@@H]1C(=O)O

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
GRM8 O00222 10/20 1.00
GRM7 Q14831 10/20 1.00
GRM2 Q14416 9/20 1.00
GRM4 Q14833 9/20 1.00
GRM3 Q14832 6/20 1.00
GRM1 Q13255 6/20 1.00
GRM5 P41594 4/20 1.00
MEN1 O00255 1/20 1.00
CYP1A2 P05177 1/20 1.00
KMT2A Q03164 1/20 1.00

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30079684 1.00 GRM8 (1.00) GRM8GRM7GRM2GRM4GRM3
SCHEMBL15060588 1.00 GRM8 (1.00) GRM8GRM7GRM2GRM4GRM3
SCHEMBL12019053 1.00 GRM8 (1.00) GRM8GRM7GRM2GRM4GRM3
SCHEMBL13746359 1.00 GRM8 (1.00) GRM8GRM7GRM2GRM4GRM3
SCHEMBL8490722 1.00 GRM8 (1.00) GRM8GRM7GRM2GRM4GRM3
SCHEMBL29389814 1.00 GRM8 (1.00) GRM8GRM7GRM2GRM4GRM3
SCHEMBL24606222 1.00 GRM8 (1.00) GRM8GRM7GRM2GRM4GRM3
SCHEMBL481153 1.00 GRM8 (1.00) GRM8GRM7GRM2GRM4GRM3
SCHEMBL7386669 0.84 GRM8 (0.72) GRM8GRM7GRM2GRM4GRM3
SCHEMBL7393500 0.84 GRM8 (0.72) GRM8GRM7GRM2GRM4GRM3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20210228508-A1 COMPOSITIONS AND METHODS THEREOF Exciva GmbH 2021-07-29 US disclosed
EP-1817300-A1 POTENTIATORS OF GLUTAMATE RECEPTORS ELI LILLY AND COMPANY (US) 2007-08-15 EP disclosed
WO-2006057860-A1 POTENTIATORS OF GLUTAMATE RECEPTORS ELI LILLY AND COMPANY (US) 2006-06-01 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20210228508-A1 COMPOSITIONS AND METHODS THEREOF CYP21A2, CYP2C19, CYP2F1 GRM8 4497/4885GRM7 3919/4885GRM2 4180/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.