SCHEMBL5202385

SCHEMBL5202385

CCOC(=O)CCCNc1ccc(Cl)cc1Oc1cccc([C@@H](C)NC(=O)OC(C)(C)C)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
MAPT P10636 3/20 0.37
KDM4E B2RXH2 2/20 0.37
ALDH1A1 P00352 2/20 0.37
GAA P10253 1/20 0.37
PKM P14618 1/20 0.37
HPGD P15428 1/20 0.37
ALOX12 P18054 1/20 0.37
PTGER4 P35408 2/20 0.36
PFKFB3 Q16875 1/20 0.36
CTSK P43235 2/20 0.36
SMN1; SMN2 Q16637 2/20 0.35
LMNA P02545 1/20 0.35
HTT P42858 1/20 0.35
PTGER2 P43116 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2D6 P10635 1/20 0.34
CYP2C19 P33261 1/20 0.34
ROCK1 Q13464 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5208051 1.00 MEN1 (0.41) MEN1KMT2AMAPTKDM4EALDH1A1
SCHEMBL5206639 0.89 KDM4E (0.36) MEN1KMT2AMAPTKDM4EPFKFB3
SCHEMBL5206633 0.84 KDM4E (0.40) MEN1KMT2AMAPTKDM4EALDH1A1
SCHEMBL5205312 0.84 PPARG (0.40) MAPTKDM4EALDH1A1SMN1; SMN2HTT
SCHEMBL5202388 0.83 CNR1 (0.40) MEN1KMT2AMAPTKDM4E
SCHEMBL5205112 0.82 MEN1 (0.37) MEN1KMT2AKDM4EALDH1A1PKM
SCHEMBL5202903 0.81 PPARG (0.40) ALDH1A1SMN1; SMN2HTTCYP3A4
SCHEMBL5208682 0.81 PPARG (0.39) CYP3A4
SCHEMBL5205300 0.78 PPARG (0.41) MEN1KMT2AKDM4EALDH1A1GAA
SCHEMBL5206532 0.78 SCN9A (0.39) MAPTKDM4EALDH1A1GAAPKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7160887-B1 Aromatic amine derivatives, their production and use TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2007-01-09 US disclosed
EP-1123918-B1 AROMATIC AMINE DERIVATIVES, PROCESS FOR THE PREPARATION THEREOF AND AGENTS CONTAINING THE SAME TAKEDA PHARMACEUTICAL (JP) 2005-03-09 EP disclosed
EP-1123918-A1 AROMATIC AMINE DERIVATIVES, PROCESS FOR THE PREPARATION THEREOF AND AGENTS CONTAINING THE SAME Takeda Chemical Industries, Ltd. (JP) 2001-08-16 EP disclosed