SCHEMBL5202471

SCHEMBL5202471

COc1ccc(-c2nc(C)c(CN)cc2-c2ccc(Cl)cc2Cl)cc1

nearest known ligand 0.55

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 14/20 0.55
DPP8 Q6V1X1 8/20 0.53
DPP9 Q86TI2 6/20 0.53
CYP3A4 P08684 1/20 0.48
CNR1 P21554 2/20 0.43
CNR2 P34972 1/20 0.43
PTPN1 P18031 1/20 0.41
CRHR1 P34998 1/20 0.41
CXCR2 P25025 1/20 0.41
MARS1 P56192 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL4912438 0.99 DPP4 (0.54) DPP4DPP8DPP9CYP3A4CNR1
SCHEMBL5189117 0.91 DPP4 (0.57) DPP4DPP8DPP9CYP3A4CNR1
SCHEMBL4934709 0.90 DPP4 (0.48) DPP4DPP8DPP9CYP3A4
Hydrochloric Acid SCHEMBL4918479 0.89 DPP4 (0.47) DPP4DPP8DPP9CYP3A4
SCHEMBL4906797 0.86 DPP4 (0.53) DPP4DPP8DPP9CYP3A4CNR1
SCHEMBL5187409 0.86 DPP4 (0.44) DPP4DPP8DPP9CRHR1
Hydrochloric Acid SCHEMBL4913608 0.85 DPP4 (0.43) DPP4DPP8DPP9CRHR1
SCHEMBL4912767 0.83 DPP4 (0.52) DPP4DPP8DPP9CYP3A4CNR1
SCHEMBL3106224 0.82 DPP4 (0.47) DPP4CNR1CNR2CRHR1
SCHEMBL4911607 0.79 HSD11B1 (0.43) DPP4DPP8DPP9CRHR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1805143-A1 PYRIDINE DERIVATIVES AND THE PREPARATION AND THE THERAPEUTIC USE THEREOF Sanofi-Aventis (FR) 2007-07-11 EP disclosed
WO-2006042955-A1 PYRIDINE DERIVATIVES AND THE PREPARATION AND THE THERAPEUTIC USE THEREOF SANOFI-AVENTIS (FR) 2006-04-27 WO disclosed