SCHEMBL5202479

SCHEMBL5202479

CCNC(=O)c1ccc2cc(C)n(C3CCN(CCc4ccc(F)cc4)CC3)c2c1

nearest known ligand 0.47

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 3/20 0.47
HTR2C P28335 2/20 0.47
HTR7 P34969 2/20 0.47
HTR6 P50406 2/20 0.47
PLD2 O14939 8/20 0.47
PLD1 Q13393 7/20 0.47
YEATS4 O95619 1/20 0.44
KCNH2 Q12809 1/20 0.44
CACNA1G O43497 1/20 0.44
DRD2 P14416 1/20 0.43
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
DRD4 P21917 1/20 0.42
CYP2D6 P10635 1/20 0.42
CHRM1 P11229 1/20 0.42
MCHR1 Q99705 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5872222 0.91 PLD2 (0.50) HTR2AHTR2CHTR7HTR6PLD2
SCHEMBL5871535 0.91 PLD2 (0.50) HTR2AHTR2CHTR7HTR6PLD2
SCHEMBL5204133 0.91 HTR2A (0.49) HTR2AHTR2CHTR7HTR6PLD2
SCHEMBL6620022 0.90 PLD2 (0.46) HTR2AHTR2CHTR7HTR6PLD2
SCHEMBL5871928 0.90 PLD2 (0.53) HTR2AHTR2CHTR7HTR6PLD2
SCHEMBL5871154 0.90 PLD2 (0.49) HTR2AHTR2CHTR7HTR6PLD2
SCHEMBL6621516 0.89 PLD2 (0.44) HTR2AHTR2CHTR7HTR6PLD2
SCHEMBL5871452 0.89 PLD2 (0.48) HTR2AHTR2CHTR7HTR6PLD2
Oxalic Acid SCHEMBL5870981 0.88 PLD2 (0.44) HTR2AHTR2CHTR7HTR6PLD2
Oxalic Acid SCHEMBL5871790 0.88 PLD2 (0.51) PLD2PLD1CACNA1GDRD2MCHR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1179532-B1 PROCESS FOR THE PRODUCTION OF INDOLE DERIVATIVES AND INTERMEDIATES THEREFOR EISAI R&D MAN CO LTD (JP) 2007-06-13 EP disclosed
US-6573384-B1 1,4-substituted cyclic amine compound which is useful as a pharmaceutical, and an intermediate for the process EISAI CO., LTD. (JP) 2003-06-03 US disclosed
EP-1179532-A1 PROCESS FOR THE PRODUCTION OF INDOLE DERIVATIVES AND INTERMEDIATES THEREFOR Eisai Co., Ltd. (JP) 2002-02-13 EP disclosed