SCHEMBL5203922

SCHEMBL5203922

CCC(=O)CCCCCC(NC(=O)Cn1ccnc1)C(=O)NCc1csc(-c2ccccc2)n1

nearest known ligand 0.42

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
PADI4 Q9UM07 1/20 0.39
ROCK2 O75116 1/20 0.38
GRK2 P25098 1/20 0.38
HPGD P15428 2/20 0.38
MGLL Q99685 1/20 0.38
TP53 P04637 1/20 0.38
KLKB1 P03952 2/20 0.37
KLK1 P06870 2/20 0.37
HDAC1 Q13547 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5117813 1.00 NPC1 (0.41) NPC1RAB9APADI4ROCK2GRK2
SCHEMBL5130351 0.84 TP53 (0.48) NPC1RAB9AHPGDTP53HDAC1
SCHEMBL5127204 0.84 HDAC1 (0.45) NPC1RAB9AHPGDTP53HDAC1
SCHEMBL5117437 0.83 NPC1 (0.46) NPC1RAB9AHPGDTP53KLK1
SCHEMBL5121951 0.83 RAB9A (0.46) NPC1RAB9AHPGDHDAC1
SCHEMBL5240614 0.83 RAB9A (0.45) NPC1RAB9AHPGDTP53HDAC1
SCHEMBL5118770 0.83 RAB9A (0.45) NPC1RAB9AHPGDTP53HDAC1
SCHEMBL5123458 0.82 RAB9A (0.44) NPC1RAB9AHPGDTP53HDAC1
SCHEMBL5131334 0.82 NPC1 (0.44) NPC1RAB9AROCK2GRK2HPGD
SCHEMBL5117937 0.82 HPGD (0.45) NPC1RAB9AHPGDTP53HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1768955-A1 AMIDE DERIVATIVES AS INHIBITORS OF HISTONE DEACETYLASE ISTITUTO DI RICERCHE DI BIOLOGIA MOLECOLARE P. ANGELETTI S.P.A. (IT) 2007-04-04 EP disclosed
WO-2006005941-A1 AMIDE DERIVATIVES AS INHIBITORS OF HISTONE DEACETYLASE ISTITUTO DI RICERCHE DI BIOLOGIA MOLECOLARE P ANGELETTI S.P.A. (IT) 2006-01-19 WO disclosed