SCHEMBL5203987

SCHEMBL5203987

Nc1cccc(OCC2=NCCN2)c1

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NISCH Q9Y2I1 11/20 0.68
MAOB P27338 4/20 0.68
MAOA P21397 3/20 0.68
HTR1A P08908 3/20 0.50
ADRA2A P08913 3/20 0.50
ADRA2B P18089 3/20 0.50
ADRA2C P18825 3/20 0.50
ADRA1A P35348 4/20 0.48
ADRA1D P25100 2/20 0.48
ADRA1B P35368 2/20 0.48
HTR1B P28222 1/20 0.48
CYP1A2 P05177 1/20 0.47
CYP2D6 P10635 1/20 0.47
THRB P10828 1/20 0.47
TSHR P16473 1/20 0.47
CYP2C19 P33261 1/20 0.47
THPO P40225 1/20 0.47
HSD17B10 Q99714 1/20 0.47
APP P05067 1/20 0.47
TP53 P04637 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL5201240 0.99 NISCH (0.66) NISCHMAOBMAOAHTR1AADRA2A
SCHEMBL3173653 0.82 NISCH (0.68) NISCHMAOBMAOAHTR1AADRA2A
SCHEMBL546875 0.81 NISCH (1.00) NISCHMAOBMAOAHTR1AADRA2A
SCHEMBL11264214 0.80 NISCH (0.68) NISCHMAOBMAOAHTR1AADRA2A
SCHEMBL11130963 0.80 NISCH (0.64) NISCHMAOBMAOAHTR1AADRA2A
SCHEMBL5203974 0.80 NISCH (0.59) NISCHMAOBMAOAHTR1AADRA2A
Hydrochloric Acid SCHEMBL11259967 0.80 NISCH (0.97) NISCHMAOBMAOAHTR1AADRA2A
SCHEMBL3172398 0.79 NISCH (0.71) NISCHMAOBMAOAHTR1AADRA2A
SCHEMBL3163279 0.79 NISCH (0.62) NISCHMAOBMAOAHTR1AADRA2A
Hydrochloric Acid SCHEMBL5201234 0.79 NISCH (0.58) NISCHMAOBMAOAHTR1AADRA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0887346-B1 N-Phenyl-alkylsulfonamide derivatives, their preparation and their use as alpha1A/1L adrenoceptor agonists HOFFMANN LA ROCHE (CH) 2007-12-12 EP disclosed
CN-1262547-C Phenyl-and aminophenyl-alkyl sulfonamide and urea derivative HOFFMANN LA ROCHE (CH) 2006-07-05 CN disclosed
CN-1176910-C Phenyl-and aminophenyl-alkylsulfonamide and urea derivatives - 2004-11-24 CN disclosed
CN-1515562-A Phenyl-and aminophenyl-alkyl sulfonamide and urea derivative - 2004-07-28 CN disclosed
CN-1515559-A Phenyl-and aminophenyl-alkyl sulfonamide and urea derivative - 2004-07-28 CN disclosed
CN-1203228-A Phenyl-and aminophenyl-alkylsulfonamide and urea derivatives HOFFMANN LA ROCHE (CH) 1998-12-30 CN disclosed
US-4523020-A USEFUL FOR TREATMENT OF DIARRHEA AND AS ANALGESICS G. D. SEARLE & CO. (US) 1985-06-11 US disclosed
US-4523020-A USEFUL FOR TREATMENT OF DIARRHEA AND AS ANALGESICS G. D. SEARLE & CO. (US) 1985-06-11 US disclosed
US-4523020-A USEFUL FOR TREATMENT OF DIARRHEA AND AS ANALGESICS G. D. SEARLE & CO. (US) 1985-06-11 US disclosed