SCHEMBL5203974

SCHEMBL5203974

NC(=O)c1cccc(OCC2=NCCN2)c1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NISCH Q9Y2I1 8/20 0.59
MAOA P21397 2/20 0.59
MAOB P27338 2/20 0.59
ADRA1A P35348 6/20 0.46
PARP1 P09874 1/20 0.46
HTR1A P08908 3/20 0.45
ADRA2A P08913 3/20 0.45
ADRA2B P18089 3/20 0.45
ADRA2C P18825 3/20 0.45
ADRA1B P35368 5/20 0.44
ADRA1D P25100 4/20 0.44
TNKS O95271 1/20 0.43
PARP15 Q460N3 1/20 0.43
PARP14 Q460N5 1/20 0.43
PARP10 Q53GL7 1/20 0.43
TNKS2 Q9H2K2 1/20 0.43
PARP2 Q9UGN5 1/20 0.43
HTR1B P28222 2/20 0.43
CYP1A2 P05177 1/20 0.42
CYP2D6 P10635 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL5201234 0.99 NISCH (0.58) NISCHMAOAMAOBADRA1APARP1
SCHEMBL5203987 0.80 NISCH (0.68) NISCHMAOAMAOBADRA1AHTR1A
Hydrochloric Acid SCHEMBL5201240 0.79 NISCH (0.66) NISCHMAOAMAOBADRA1AHTR1A
SCHEMBL11264214 0.77 NISCH (0.68) NISCHMAOAMAOBADRA1AHTR1A
SCHEMBL3173653 0.77 NISCH (0.68) NISCHMAOAMAOBADRA1AHTR1A
SCHEMBL546875 0.76 NISCH (1.00) NISCHMAOAMAOBADRA1AHTR1A
SCHEMBL11270249 0.75 NISCH (0.61) NISCHMAOAMAOBHTR1AADRA2A
SCHEMBL11130963 0.75 NISCH (0.64) NISCHMAOAMAOBADRA1AHTR1A
Hydrochloric Acid SCHEMBL11259967 0.74 NISCH (0.97) NISCHMAOAMAOBADRA1AHTR1A
SCHEMBL3163279 0.74 NISCH (0.62) NISCHMAOAMAOBADRA1AHTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0887346-B1 N-Phenyl-alkylsulfonamide derivatives, their preparation and their use as alpha1A/1L adrenoceptor agonists HOFFMANN LA ROCHE (CH) 2007-12-12 EP disclosed
CN-1262547-C Phenyl-and aminophenyl-alkyl sulfonamide and urea derivative HOFFMANN LA ROCHE (CH) 2006-07-05 CN disclosed
CN-1176910-C Phenyl-and aminophenyl-alkylsulfonamide and urea derivatives - 2004-11-24 CN disclosed
CN-1515562-A Phenyl-and aminophenyl-alkyl sulfonamide and urea derivative - 2004-07-28 CN disclosed
CN-1515559-A Phenyl-and aminophenyl-alkyl sulfonamide and urea derivative - 2004-07-28 CN disclosed
CN-1203228-A Phenyl-and aminophenyl-alkylsulfonamide and urea derivatives HOFFMANN LA ROCHE (CH) 1998-12-30 CN disclosed