SCHEMBL5204879

SCHEMBL5204879

Nc1cccc2c1C(=O)NS2(=O)=O

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RET P07949 2/20 0.62
GRK5 P34947 2/20 0.62
TYRO3 Q06418 2/20 0.62
DYRK1B Q9Y463 2/20 0.62
CA12 O43570 14/20 0.50
CA9 Q16790 14/20 0.50
CA2 P00918 13/20 0.50
CA1 P00915 11/20 0.50
CA7 P43166 10/20 0.50
CA4 P22748 9/20 0.50
KDM4E B2RXH2 2/20 0.50
USP2 O75604 1/20 0.50
LMNA P02545 1/20 0.50
BCHE P06276 1/20 0.50
CA6 P23280 1/20 0.50
CA5A P35218 1/20 0.50
KMT2A Q03164 1/20 0.50
CA14 Q9ULX7 1/20 0.50
CA5B Q9Y2D0 1/20 0.50
PTPRC P08575 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30834818 1.00 RET (0.62) RETGRK5TYRO3DYRK1BCA12
SCHEMBL7023285 0.81 RET (0.62) RETGRK5TYRO3DYRK1BCA12
SCHEMBL1725776 0.77 RET (1.00) RETGRK5TYRO3DYRK1BCA12
SCHEMBL3961225 0.77 RET (0.62) RETGRK5TYRO3DYRK1BCA12
SCHEMBL7381362 0.77 RET (0.62) RETGRK5TYRO3DYRK1BCA12
SCHEMBL9620282 0.77 RET (0.62) RETGRK5TYRO3DYRK1BCA12
SCHEMBL11155230 0.76 RET (0.61) RETGRK5TYRO3DYRK1BCA12
SCHEMBL7287038 0.75 RET (0.56) RETGRK5TYRO3DYRK1BCA12
SCHEMBL7778266 0.74 RET (0.46) RETGRK5TYRO3DYRK1BCA12
SCHEMBL7280743 0.74 RET (0.59) RETGRK5TYRO3DYRK1BCA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 46 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6776930-B2 POLYMER BONDED TO DYE EASTMAN KODAK COMPANY 2004-08-17 US claimed
US-20010023938-A1 Polymer bonded to dye ALLEN MAX (US) 2001-09-27 US claimed
US-6197223-B1 REACTING DIACIDIC MONOMER HAVING FORMULA H--A--H, COMPRISING 1 TO 100 MOLE % OF LIGHT-ABSORBING MONOMER HAVING A LIGHT ABSORPTION MAXIMUM BETWEEN 300 NM AND 1200 NM AND 99-0 MOLE % OF A NON-LIGHT ABSORBING MONOMER WITH ORGANIC COMPOUND EASTMAN CHEMICAL COMPANY 2001-03-06 US claimed
EP-0948570-A1 METHOD FOR PREPARING LIGHT-ABSORBING POLYMERIC COMPOSITIONS EASTMAN CHEMICAL COMPANY (US) 1999-10-13 EP claimed
WO-1998023690-A9 METHOD FOR PREPARING LIGHT-ABSORBING POLYMERIC COMPOSITIONS 1998-09-17 WO claimed
WO-1998023690-A1 METHOD FOR PREPARING LIGHT-ABSORBING POLYMERIC COMPOSITIONS EASTMAN CHEMICAL COMPANY (US) 1998-06-04 WO claimed
US-20230353959-A1 PI3K-ALPHA INHIBITORS AND METHODS OF USE THEREOF RELAY THERAPEUTICS, INC. 2023-11-02 US disclosed
CN-116261562-A PI 3K-alpha inhibitors and methods of use thereof 传达治疗有限公司 2023-06-13 CN disclosed
WO-2021222556-A1 PI3K-α INHIBITORS AND METHODS OF USE THEREOF RELAY THERAPEUTICS, INC. (US) 2021-11-04 WO disclosed
EP-1739135-A2 Colorant compounds containing copolymerizable vinyl groups Eastman Chemical Company (US) 2007-01-03 EP disclosed
EP-1307515-B1 COLORANT COMPOUNDS CONTAINING COPOLYMERIZABLE VINYL GROUPS EASTMAN CHEM CO (US) 2006-06-28 EP disclosed
US-7060829-B2 Colorant compounds containing copolymerizable vinyl groups EASTMAN CHEMICAL COMPANY (US) 2006-06-13 US disclosed
US-7030244-B2 Colorant compounds containing copolymerizable vinyl groups EASTMAN CHEMICAL COMPANY (US) 2006-04-18 US disclosed
EP-0550112-A1 2-Saccharinylmethyl aryl and aryloxy acetates useful as proteolytic enzyme inhibitors and pharmaceutical compositions contaning them STERLING WINTHROP INC. (US) 1993-07-07 EP disclosed
EP-0549073-A1 Novel 2-saccharinylmethyl and 4,5,6,7-tetrahydro-2-saccharinylmethyl phosphates, phosphonates and phosphinates useful as proteolytic enzyme inhibitors and compositions and method of use thereof STERLING WINTHROP INC. (US) 1993-06-30 EP disclosed
US-5187173-A Degenerative diseases such as emphysema, rheumatoid arthritis, pancreatitis, cyctic fibrosis and skin disorders STERLING WINTHROP INC. (US) 1993-02-16 US disclosed
US-5128339-A Emphysema, rheumatoid arthritis, pancreatitis STERLING WINTHROP INC. (US) 1992-07-07 US disclosed
EP-0483928-A1 2-Saccharinylmethyl aryl carboxylates useful as proteolytic enzyme inhibitors and compositions and method of use STERLING WINTHROP INC. (US) 1992-05-06 EP disclosed
US-4404230-A ARTICIFIAL SWEETENERS DR. KARL THOMAE GMBH (DE) 1983-09-13 US disclosed
US-3878189-A Azo dye compounds from amino-1,2-benzisothiazolon-1,1-dioxides CIBA-GEIGY CORPORATION, A CORP. OF NEW YORK 1975-04-15 US disclosed