SCHEMBL5205141

SCHEMBL5205141

O=C(c1ccccc1Cl)N1CCC(c2c[nH]c3ccccc23)C1

nearest known ligand 0.63

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 7/20 0.63
KDM4E B2RXH2 3/20 0.60
ALDH1A1 P00352 2/20 0.60
BRD4 O60885 1/20 0.60
POLB P06746 1/20 0.60
CREBBP Q92793 1/20 0.60
ATM Q13315 1/20 0.54
RAB9A P51151 1/20 0.50
CCR2 P41597 2/20 0.49
CYP2D6 P10635 1/20 0.48
GAA P10253 1/20 0.47
AVPR1A P37288 1/20 0.47
ADRA1D P25100 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5202689 0.81 HSD11B1 (0.67) HSD11B1KDM4EALDH1A1BRD4POLB
SCHEMBL16801592 0.81 KDM4E (0.85) HSD11B1KDM4EALDH1A1BRD4POLB
SCHEMBL13666115 0.78 HSD11B1 (0.59) HSD11B1KDM4EALDH1A1BRD4POLB
SCHEMBL19248198 0.77 HSD11B1 (1.00) HSD11B1KDM4EALDH1A1BRD4POLB
SCHEMBL16801846 0.77 KDM4E (0.74) HSD11B1KDM4EALDH1A1BRD4POLB
SCHEMBL5705116 0.76 KDM4E (0.78) HSD11B1KDM4EALDH1A1BRD4POLB
SCHEMBL27201572 0.76 HSD11B1 (0.64) HSD11B1KDM4EALDH1A1BRD4POLB
SCHEMBL16801703 0.76 KDM4E (0.72) HSD11B1KDM4EALDH1A1BRD4POLB
SCHEMBL18324984 0.75 KDM4E (0.76) HSD11B1KDM4EALDH1A1BRD4POLB
SCHEMBL5705098 0.75 KDM4E (1.00) HSD11B1KDM4EALDH1A1BRD4POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1654253-B1 SUBSTITUTED 3-PYRROLIDIN-INDOLE DERIVATIVES GRUENENTHAL GMBH (DE) 2007-01-03 EP claimed
EP-1654253-B1 SUBSTITUTED 3-PYRROLIDIN-INDOLE DERIVATIVES GRUENENTHAL GMBH (DE) 2007-01-03 EP disclosed