SCHEMBL5205314

SCHEMBL5205314

NCc1cccc(Oc2ccccc2N)c1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.60
ALDH1A1 P00352 1/20 0.60
RCE1 Q9Y256 1/20 0.54
F10 P00742 1/20 0.45
TLR4 O00206 1/20 0.44
DPP4 P27487 1/20 0.44
LOXL2 Q9Y4K0 3/20 0.43
KDM4E B2RXH2 1/20 0.42
MAPT P10636 1/20 0.42
CRHBP P24387 1/20 0.42
CRHR2 Q13324 1/20 0.42
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
MAOB P27338 1/20 0.41
IKBKB O14920 1/20 0.41
BRAF P15056 1/20 0.41
LOX P28300 1/20 0.41
NOS1 P29475 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13452511 0.85 GAA (0.58) GAAALDH1A1RCE1F10TLR4
SCHEMBL1049509 0.83 ALDH1A1 (0.75) GAAALDH1A1RCE1F10TLR4
SCHEMBL921481 0.81 DPP4 (0.58) GAAALDH1A1F10DPP4LOXL2
SCHEMBL922401 0.81 FFAR1 (0.51) GAAALDH1A1F10DPP4LOXL2
SCHEMBL922873 0.81 F10 (0.50) F10DPP4LOXL2MAOBLOX
SCHEMBL921026 0.81 ALDH1A1 (0.53) GAAALDH1A1F10KDM4EMAOB
Ammonia Solution, Strong SCHEMBL10884991 0.81 ALDH1A1 (0.72) GAAALDH1A1RCE1F10TLR4
SCHEMBL6289782 0.81 ALDH1A1 (0.72) GAAALDH1A1RCE1F10TLR4
SCHEMBL6290404 0.81 ALDH1A1 (0.72) GAAALDH1A1RCE1F10TLR4
SCHEMBL1270999 0.81 ALDH1A1 (0.72) GAAALDH1A1RCE1F10TLR4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7160887-B1 Aromatic amine derivatives, their production and use TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2007-01-09 US disclosed
EP-1123918-B1 AROMATIC AMINE DERIVATIVES, PROCESS FOR THE PREPARATION THEREOF AND AGENTS CONTAINING THE SAME TAKEDA PHARMACEUTICAL (JP) 2005-03-09 EP disclosed
EP-1123918-A1 AROMATIC AMINE DERIVATIVES, PROCESS FOR THE PREPARATION THEREOF AND AGENTS CONTAINING THE SAME Takeda Chemical Industries, Ltd. (JP) 2001-08-16 EP disclosed