SCHEMBL5205748

SCHEMBL5205748

NC(=O)Nc1ccc2c(c1)CCC2

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 14/20 0.63
RAB9A P51151 14/20 0.63
MEN1 O00255 1/20 0.63
KMT2A Q03164 1/20 0.63
SMN1; SMN2 Q16637 5/20 0.61
POLB P06746 3/20 0.61
NFKB1 P19838 3/20 0.61
NFKB2 Q00653 3/20 0.61
RELA Q04206 3/20 0.61
TP53 P04637 2/20 0.61
GAA P10253 1/20 0.61
HTT P42858 1/20 0.61
CA12 O43570 1/20 0.59
CA1 P00915 1/20 0.59
CA2 P00918 1/20 0.59
CA9 Q16790 1/20 0.59
MAPT P10636 2/20 0.58
ALDH1A1 P00352 1/20 0.58
LY96 Q9Y6Y9 1/20 0.58
PLAU P00749 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8884002 0.98 NPC1 (0.61) NPC1RAB9AMEN1KMT2ASMN1; SMN2
SCHEMBL12539916 0.84 MELK (0.61) NPC1RAB9AMEN1KMT2ASMN1; SMN2
SCHEMBL11896022 0.83 NPC1 (0.70) NPC1RAB9AMEN1KMT2ASMN1; SMN2
SCHEMBL4072601 0.83 HTR1A (0.52) NPC1RAB9AMEN1KMT2ASMN1; SMN2
SCHEMBL7837810 0.82 BAZ2B (0.73)
SCHEMBL3771009 0.81 PLAU (0.57) NPC1RAB9AMEN1KMT2ASMN1; SMN2
SCHEMBL1673429 0.81 BAZ2B (0.69) NPC1RAB9AMEN1KMT2ASMN1; SMN2
SCHEMBL1878955 0.81 PTPN7 (0.57) NPC1RAB9AMEN1KMT2ASMN1; SMN2
SCHEMBL30494024 0.79 NPC1 (0.65) NPC1RAB9AMEN1KMT2ASMN1; SMN2
SCHEMBL20119168 0.79 TMPRSS2 (0.50) CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1023072-A1 ANALGESIC COMPOSITIONS Panos Therapeutics Limited (GB) 2000-08-02 EP claimed
WO-1999018967-A1 ANALGESIC COMPOSITIONS PANOS THERAPEUTICS LIMITED (GB) 1999-04-22 WO claimed
US-5696110-A ANTIULCER AGENTS MERCK, SHARP & DOHME, LTD. (GB) 1997-12-09 US claimed
EP-0652871-A1 BENZODIAZEPINE DERIVATIVES MERCK SHARP & DOHME LTD. (GB) 1995-05-17 EP claimed
EP-1804785-A2 DIARYL UREAS AS CB1 ANTAGONISTS NEUROGEN CORPORATION (US) 2007-07-11 EP disclosed
WO-2006049941-A2 DIARYL UREAS AS CB1 ANTAGONISTS NEUROGEN CORPORATION (US) 2006-05-11 WO disclosed
US-5696110-A ANTIULCER AGENTS MERCK, SHARP & DOHME, LTD. (GB) 1997-12-09 US disclosed
US-5663331-A BACTERICIDES IL-DONG PHARM. CO., LTD. (KR) 1997-09-02 US disclosed
WO-1993015084-A1 NOVEL CEPHALOSPORIN COMPOUNDS IL-DONG PHARM. CO., LTD. (KR) 1993-08-05 WO disclosed