SCHEMBL5206410

SCHEMBL5206410

CC(C)(C)c1ccc(CCNCCc2cccc(C(F)(F)F)c2)cc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 1/20 0.51
KDM4E B2RXH2 2/20 0.51
TDP1 Q9NUW8 1/20 0.51
MEN1 O00255 1/20 0.50
KMT2A Q03164 1/20 0.50
ROCK1 Q13464 1/20 0.48
HDAC1 Q13547 1/20 0.48
HDAC8 Q9BY41 1/20 0.48
SIGMAR1 Q99720 2/20 0.47
TP53 P04637 1/20 0.47
CYP1A2 P05177 1/20 0.47
CYP3A4 P08684 1/20 0.47
CYP2D6 P10635 1/20 0.47
TSHR P16473 1/20 0.47
CYP2C19 P33261 1/20 0.47
HTR2A P28223 2/20 0.45
HTR2B P41595 2/20 0.45
HTR2C P28335 1/20 0.45
MIF P14174 1/20 0.44
CNR1 P21554 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3235999 0.92 KDM4E (0.58) TAAR1KDM4ETDP1MEN1KMT2A
SCHEMBL12521121 0.83 SCN8A (0.54) TAAR1KDM4ETDP1MEN1KMT2A
SCHEMBL10562876 0.83 TAAR1 (0.56) TAAR1KDM4ETDP1MEN1KMT2A
Hydrochloric Acid SCHEMBL10560147 0.82 TAAR1 (0.54) TAAR1KDM4ETDP1MEN1KMT2A
SCHEMBL18161368 0.81 TAAR1 (0.65) TAAR1KDM4EHDAC1HDAC8SIGMAR1
SCHEMBL5175432 0.80 KDM4E (0.49) TAAR1KDM4ETDP1MEN1KMT2A
SCHEMBL5176778 0.80 KDM4E (0.49) TAAR1KDM4ETDP1MEN1KMT2A
SCHEMBL5175308 0.80 KDM4E (0.55) TAAR1KDM4ETDP1MEN1KMT2A
SCHEMBL5177801 0.80 ADRA2C (0.52) TAAR1KDM4EMEN1KMT2ASIGMAR1
SCHEMBL28246680 0.79 TAAR1 (0.55) TAAR1KDM4ETDP1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1776338-A1 INDOLE, INDAZOLE OR INDOLINE DERIVATIVES F. Hoffmann-Roche AG (CH) 2007-04-25 EP disclosed
WO-2006013048-A1 INDOLE, INDAZOLE OR INDOLINE DERIVATIVES F.HOFFMANN-LA ROCHE AG (CH) 2006-02-09 WO disclosed