SCHEMBL5207438

SCHEMBL5207438

Cn1cc(-c2nc(-c3ccc(Cl)cc3)c(CCC(=O)N3CCS(=O)(=O)CC3)o2)c2ccccc21

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.40
LMNA P02545 2/20 0.40
POLB P06746 2/20 0.40
MAPK1 P28482 1/20 0.40
HTT P42858 1/20 0.40
ALDH1A1 P00352 3/20 0.40
KDM4E B2RXH2 2/20 0.40
NPSR1 Q6W5P4 2/20 0.40
HSD17B10 Q99714 1/20 0.40
TNKS O95271 1/20 0.36
PARP1 P09874 1/20 0.36
PARP2 Q9UGN5 1/20 0.36
NPC1 O15118 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36
HPGD P15428 1/20 0.36
RAB9A P51151 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
TACR1 P25103 4/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5209815 0.89 TACR1 (0.41) MAPTLMNAPOLBMAPK1HTT
SCHEMBL5214208 0.86 TACR1 (0.46) MAPTLMNAPOLBMAPK1HTT
SCHEMBL5210928 0.84 RXRA (0.46) ALDH1A1KDM4ENPC1CYP1A2CYP3A4
SCHEMBL5214817 0.82 KDM4E (0.40) MAPTLMNAPOLBHTTALDH1A1
SCHEMBL5209029 0.78 POLB (0.47) MAPTLMNAPOLBMAPK1HTT
SCHEMBL5210227 0.78 POLB (0.41) MAPTLMNAPOLBMAPK1HTT
SCHEMBL5209589 0.76 POLB (0.50) MAPTLMNAPOLBMAPK1HTT
SCHEMBL5211815 0.76 POLB (0.47) MAPTLMNAPOLBMAPK1HTT
SCHEMBL5210396 0.76 MEN1 (0.43) MAPTLMNAPOLBHTTALDH1A1
SCHEMBL5207233 0.75 POLB (0.37) MAPTPOLBTNKSPARP1PARP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7183276-B2 Azole compounds TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2007-02-27 US claimed
US-7183276-B2 Azole compounds TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2007-02-27 US disclosed