SCHEMBL5207693

SCHEMBL5207693

C=CCOc1ccc(S(C)(=O)=O)cc1Oc1ccccc1

nearest known ligand 0.49

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 2/20 0.47
PTGDR2 Q9Y5Y4 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.41
CA12 O43570 1/20 0.41
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
CA7 P43166 1/20 0.41
CA9 Q16790 1/20 0.41
BRD4 O60885 3/20 0.40
SLC6A4 P31645 1/20 0.39
KCNQ3 O43525 5/20 0.39
KCNQ2 O43526 5/20 0.39
NPSR1 Q6W5P4 1/20 0.38
KCNQ5 Q9NR82 2/20 0.38
KCNQ4 P56696 1/20 0.38
PTGS1 P23219 1/20 0.38
KDM4E B2RXH2 1/20 0.38
GAA P10253 1/20 0.37
TSHR P16473 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5757380 0.85 PTGS2 (0.50) PTGS2SMN1; SMN2CA12CA1CA2
SCHEMBL5239038 0.76 TSHR (0.49) CA12CA1CA9SLC6A4KDM4E
SCHEMBL31388364 0.75 ERN1 (0.43) PTGDR2SMN1; SMN2CA12CA1CA2
SCHEMBL5207689 0.74 CA12 (0.63) SMN1; SMN2CA12CA1CA2CA7
SCHEMBL31388318 0.74 CA12 (0.44) PTGDR2SMN1; SMN2CA12CA1CA2
SCHEMBL28745794 0.74 HPGD (0.40) PTGS2SMN1; SMN2CA12CA1CA2
SCHEMBL28623953 0.73 CA12 (0.40) PTGDR2SMN1; SMN2CA12CA1CA2
SCHEMBL15068183 0.73 PTGS2 (0.55) PTGS2PTGDR2SMN1; SMN2BRD4SLC6A4
SCHEMBL21190753 0.73 EPAS1 (0.60) PTGS2PTGDR2SMN1; SMN2BRD4PTGS1
SCHEMBL15067760 0.73 SMN1; SMN2 (0.66) PTGS2SMN1; SMN2BRD4PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1040102-B1 ARYLTHIAZOLIDINEDIONE DERIVATIVES MERCK & CO INC (US) 2007-01-24 EP disclosed
EP-1040102-A4 ARYLTHIAZOLIDINEDIONE DERIVATIVES MERCK & CO INC (US) 2002-11-27 EP disclosed
EP-1040102-A1 ARYLTHIAZOLIDINEDIONE DERIVATIVES Merck & Co., Inc. (US) 2000-10-04 EP disclosed
WO-1999032465-A1 ARYLTHIAZOLIDINEDIONE DERIVATIVES MERCK & CO., INC. (US) 1999-07-01 WO disclosed