SCHEMBL5208968

SCHEMBL5208968

CNC1CCOCC1.Cc1ccc(NC(=O)C=Cc2ccc(-c3ccc(C)cc3)s2)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCR2 P41597 3/20 0.48
LMNA P02545 4/20 0.48
MAPT P10636 4/20 0.48
MEN1 O00255 3/20 0.48
KMT2A Q03164 3/20 0.48
HTT P42858 3/20 0.48
NPC1 O15118 1/20 0.48
MMP1 P03956 4/20 0.40
MMP2 P08253 4/20 0.40
MMP9 P14780 4/20 0.40
EGFR P00533 1/20 0.40
ESRRG P62508 1/20 0.39
TRPV1 Q8NER1 1/20 0.39
TP53 P04637 2/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
RAB9A P51151 1/20 0.39
CA2 P00918 2/20 0.39
CA9 Q16790 2/20 0.39
CA12 O43570 1/20 0.39
NMT1 P30419 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7933310 0.94 CCR2 (0.44) CCR2LMNAMAPTMEN1KMT2A
SCHEMBL5208975 0.82 CCR2 (0.50) CCR2LMNAMAPTMEN1KMT2A
SCHEMBL5208961 0.82 CCR2 (0.50) CCR2LMNAMAPTMEN1KMT2A
Iodide SCHEMBL5206286 0.82 CCR2 (0.73) CCR2
Iodide SCHEMBL5206291 0.82 CCR2 (0.73) CCR2
SCHEMBL7681268 0.73 CCR2 (0.46) CCR2MAPTMEN1KMT2ATRPV1
SCHEMBL7681272 0.73 CCR2 (0.46) CCR2MAPTMEN1KMT2ATRPV1
SCHEMBL7682396 0.73 MAPK1 (0.49) CCR2LMNAMAPTNPC1EGFR
SCHEMBL7682398 0.73 MAPK1 (0.49) CCR2LMNAMAPTNPC1EGFR
SCHEMBL19003304 0.73 ABL1 (0.58) LMNAMAPTMEN1KMT2ANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1040103-B1 ANILIDE DERIVATIVE, PRODUCTION AND USE THEREOF TAKEDA PHARMACEUTICAL (JP) 2007-03-14 EP disclosed
US-6268354-B1 Pharmaceutical composition for antagonizing CCR5 comprising anilide derivative TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-07-31 US disclosed