SCHEMBL5209375

SCHEMBL5209375

CCOc1ccc(-c2ccc3c(c2)C=C(C(=O)Nc2ccc(CN(C)C4CCOCC4)cc2)CCN3C)cc1

nearest known ligand 0.60

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CCR2 P41597 5/20 0.60
CCR5 P51681 14/20 0.55
CXCR3 P49682 3/20 0.42
CCR7 P32248 2/20 0.42
MEN1 O00255 1/20 0.42
ALDH1A1 P00352 1/20 0.42
TP53 P04637 1/20 0.42
CYP1A2 P05177 1/20 0.42
CYP3A4 P08684 1/20 0.42
GAA P10253 1/20 0.42
MAPT P10636 1/20 0.42
CYP2C19 P33261 1/20 0.42
KMT2A Q03164 1/20 0.42
MCL1 Q07820 1/20 0.42
CACNA1B Q00975 1/20 0.42
APBA1 Q02410 1/20 0.42
SAE1 Q9UBE0 1/20 0.42
UBA2 Q9UBT2 1/20 0.42
CXCR5 P32302 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6351993 0.94 CCR2 (0.58) CCR2CCR5CXCR3CCR7
SCHEMBL6343858 0.94 CCR2 (0.58) CCR2CCR5CCR7
SCHEMBL6351851 0.94 CCR2 (0.58) CCR2CCR5CXCR3CCR7
SCHEMBL5209291 0.92 CCR2 (0.64) CCR2CCR5CXCR3CCR7CXCR5
SCHEMBL6343762 0.92 CCR2 (0.56) CCR2CCR5CCR7
SCHEMBL6343597 0.92 CCR2 (0.56) CCR2CCR5CCR7
SCHEMBL6342915 0.91 CCR2 (0.58) CCR2CCR5CXCR3CCR7MEN1
SCHEMBL5209524 0.90 CCR2 (0.73) CCR2CCR5CXCR3CCR7
SCHEMBL6349106 0.90 CCR2 (0.57) CCR2CCR5CXCR3CCR7MEN1
SCHEMBL5209677 0.90 CCR2 (0.58) CCR2CCR5CXCR3CCR7CXCR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1040103-B1 ANILIDE DERIVATIVE, PRODUCTION AND USE THEREOF TAKEDA PHARMACEUTICAL (JP) 2007-03-14 EP disclosed
US-6413947-B1 Anilide derivative, production and use thereof TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2002-07-02 US disclosed
US-6268354-B1 Pharmaceutical composition for antagonizing CCR5 comprising anilide derivative TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-07-31 US disclosed
US-6172061-B1 AIDS THERAPY TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-01-09 US disclosed
US-6166006-A Anilide derivative, production and use thereof TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2000-12-26 US disclosed