SCHEMBL5210446

SCHEMBL5210446

COCCOc1ccc(-c2cc3cc(NC(=O)OC(C)C)ccc3[nH]2)cc1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNQ2 O43526 1/20 0.59
NPC1 O15118 5/20 0.45
RAB9A P51151 5/20 0.45
RXFP1 Q9HBX9 1/20 0.45
CYP1A2 P05177 1/20 0.44
CYP2D6 P10635 1/20 0.44
CYP2C9 P11712 1/20 0.44
HPGD P15428 1/20 0.44
CYP2C19 P33261 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
HDAC6 Q9UBN7 1/20 0.41
L3MBTL1 Q9Y468 2/20 0.41
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
KDM4E B2RXH2 4/20 0.40
ALDH1A1 P00352 2/20 0.40
PRNP P04156 1/20 0.40
GAA P10253 1/20 0.40
MAPT P10636 2/20 0.40
NAMPT P43490 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5211787 0.85 KCNQ2 (0.62) KCNQ2NPC1RAB9ARXFP1HPGD
SCHEMBL2981789 0.85 KIT (0.49) KCNQ2HDAC6
SCHEMBL5202815 0.83 KCNQ2 (0.61) KCNQ2NPC1RAB9ASMN1; SMN2MEN1
SCHEMBL5191194 0.82 MAPT (0.49) NPC1RAB9ACYP1A2CYP2D6CYP2C9
SCHEMBL5210856 0.82 KCNQ2 (0.55) KCNQ2NPC1RAB9ACYP1A2CYP2D6
SCHEMBL2878635 0.77 NPC1 (0.60) KCNQ2NPC1RAB9ACYP1A2CYP2D6
SCHEMBL2980544 0.75 KIT (0.49)
SCHEMBL2988206 0.74 BTK (0.43) NPC1RAB9ACYP1A2CYP2D6CYP2C9
SCHEMBL2980356 0.74 KIT (0.46) KCNQ2SMN1; SMN2HDAC6
SCHEMBL2984996 0.72 KCNQ2 (0.57) KCNQ2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1831218-A2 CARBAMATE SUBSTITUTED IMIDAZO- AND PYRROLO-PYRIDINES AS PROTEIN KINASE INHIBITORS F.HOFFMANN-LA ROCHE AG (CH) 2007-09-12 EP claimed
WO-2006066914-A2 CARBAMATE SUBSTITUTED IMIDAZO- AND PYRROLO-PYRIDINES AS PROTEIN KINASE INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2006-06-29 WO claimed