SCHEMBL5202815

SCHEMBL5202815

COCCOc1ccc(-c2cc3cc(NC(=O)OCc4ccccc4)ccc3[nH]2)cc1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNQ2 O43526 1/20 0.61
TP53 P04637 2/20 0.47
MAPT P10636 2/20 0.47
NPC1 O15118 2/20 0.46
RAB9A P51151 2/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
ROCK2 O75116 2/20 0.46
MGLL Q99685 2/20 0.45
NAMPT P43490 1/20 0.45
LMNA P02545 1/20 0.44
ITGB3 P05106 1/20 0.44
ITGAV P06756 1/20 0.44
ADORA2B P29275 4/20 0.44
ADORA2A P29274 3/20 0.44
ADORA3 P0DMS8 2/20 0.44
ADORA1 P30542 2/20 0.44
JAK2 O60674 1/20 0.42
EGFR P00533 1/20 0.42
CSF1R P07333 1/20 0.42
ENPP2 Q13822 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2977727 0.86 KIT (0.51) KCNQ2TP53MAPTNPC1RAB9A
SCHEMBL5200855 0.86 MGLL (0.60) KCNQ2TP53MAPTNPC1RAB9A
SCHEMBL5211787 0.84 KCNQ2 (0.62) KCNQ2TP53MAPTNPC1RAB9A
SCHEMBL5210446 0.83 KCNQ2 (0.59) KCNQ2TP53MAPTNPC1RAB9A
SCHEMBL7908588 0.81 KCNQ2 (0.57) KCNQ2TP53MAPTNPC1RAB9A
SCHEMBL2981606 0.78 KIT (0.49) MGLLJAK2ENPP2
SCHEMBL8985906 0.74 SRD5A2 (0.60) TP53MAPTNPC1RAB9ASMN1; SMN2
SCHEMBL5272080 0.74 KCNQ2 (0.60) KCNQ2MAPTNPC1RAB9ASMN1; SMN2
SCHEMBL2984996 0.73 KCNQ2 (0.57) KCNQ2ADORA2BADORA2A
SCHEMBL8985820 0.72 MMP13 (0.68) KCNQ2TP53MAPTNPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1831218-A2 CARBAMATE SUBSTITUTED IMIDAZO- AND PYRROLO-PYRIDINES AS PROTEIN KINASE INHIBITORS F.HOFFMANN-LA ROCHE AG (CH) 2007-09-12 EP claimed
WO-2006066914-A2 CARBAMATE SUBSTITUTED IMIDAZO- AND PYRROLO-PYRIDINES AS PROTEIN KINASE INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2006-06-29 WO claimed