SCHEMBL5213183

SCHEMBL5213183

CC(C)N1CCC(OC2CCN(c3ccc(C(F)(F)F)nc3)CC2)CC1

nearest known ligand 0.61

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 12/20 0.61
CYP3A4 P08684 2/20 0.47
DHFR P00374 1/20 0.44
SLC6A9 P48067 1/20 0.43
NR1H2 P55055 1/20 0.40
NR1H3 Q13133 1/20 0.40
LCAT P04180 2/20 0.39
CHRM4 P08173 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL5214840 0.99 HRH3 (0.60) HRH3CYP3A4DHFRSLC6A9NR1H2
SCHEMBL5211308 0.85 HRH3 (0.44) HRH3SLC6A9LCAT
SCHEMBL5211979 0.81 HRH3 (0.48) HRH3SLC6A9
Hydrochloric Acid SCHEMBL5215054 0.81 HRH3 (0.47) HRH3SLC6A9
SCHEMBL5212095 0.81 HRH3 (0.48) HRH3CYP3A4DHFRLCATCHRM4
Hydrochloric Acid SCHEMBL5210871 0.80 HRH3 (0.47) HRH3CYP3A4DHFRLCATCHRM4
SCHEMBL3859666 0.79 HRH3 (0.92) HRH3CYP3A4SLC6A9CHRM4
SCHEMBL5209950 0.79 HRH3 (0.48) HRH3SLC6A9
Hydrochloric Acid SCHEMBL3878761 0.78 HRH3 (0.90) HRH3CYP3A4SLC6A9CHRM4
SCHEMBL5212466 0.78 HRH3 (0.48) HRH3LCAT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1646620-B1 SUBSTITUTED PIPERIDINES AS HISTAMINE H3 RECEPTOR LIGANDS GLAXO GROUP LTD (GB) 2007-08-15 EP claimed
EP-1646620-B1 SUBSTITUTED PIPERIDINES AS HISTAMINE H3 RECEPTOR LIGANDS GLAXO GROUP LTD (GB) 2007-08-15 EP disclosed