SCHEMBL5213635

SCHEMBL5213635

COc1cccc(CCNC(=O)C2CCCN2)c1

nearest known ligand 0.60

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.53
HTR2C P28335 2/20 0.53
HTR2B P41595 2/20 0.53
RAB9A P51151 1/20 0.52
MTNR1A P48039 2/20 0.51
MTNR1B P49286 2/20 0.51
CNR1 P21554 1/20 0.50
ALDH1A1 P00352 2/20 0.49
POLB P06746 1/20 0.49
CHRM2 P08172 1/20 0.49
CHRM1 P11229 1/20 0.49
CHRM3 P20309 1/20 0.49
CA1 P00915 1/20 0.48
CA2 P00918 1/20 0.48
CA7 P43166 1/20 0.48
CA9 Q16790 1/20 0.48
CA14 Q9ULX7 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21540797 0.85 HTR2C (0.57) KDM4EHTR2CHTR2BALDH1A1POLB
SCHEMBL13570736 0.83 CCNA2 (0.50) KDM4EHTR2CHTR2BPOLB
SCHEMBL21540592 0.82 KDM4E (0.76) KDM4EALDH1A1CA1CA2CA9
SCHEMBL21540800 0.82 TAAR1 (0.63) KDM4EHTR2CHTR2BRAB9ACNR1
SCHEMBL2089855 0.81 HTR2C (0.60) HTR2CHTR2BRAB9AALDH1A1POLB
SCHEMBL2089398 0.81 HTR2C (0.60) HTR2CHTR2BRAB9AALDH1A1POLB
SCHEMBL2089397 0.81 HTR2C (0.60) HTR2CHTR2BRAB9AALDH1A1POLB
Hydrochloric Acid SCHEMBL11095820 0.80 HTR2C (0.59) HTR2CHTR2BRAB9AALDH1A1POLB
SCHEMBL5193856 0.79 KDM4E (0.55) KDM4ERAB9AMTNR1AMTNR1BCNR1
SCHEMBL24322439 0.77 TAAR1 (0.62) KDM4EHTR2CHTR2BRAB9AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0968206-B8 N-HETEROCYCLIC DERIVATIVES AS NOS INHIBITORS BERLEX INC (US) 2007-01-24 EP disclosed
EP-0968206-A1 N-HETEROCYCLIC DERIVATIVES AS NOS INHIBITORS BERLEX LABORATORIES, INC. (US) 2000-01-05 EP disclosed
WO-1998037079-A1 N-HETEROCYCLIC DERIVATIVES AS NOS INHIBITORS BERLEX LABORATORIES, INC. (US) 1998-08-27 WO disclosed