SCHEMBL5193856

SCHEMBL5193856

COc1cccc(CCNC(=O)CC2CCCCN2)c1

nearest known ligand 0.60

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.55
ALDH1A1 P00352 2/20 0.55
CA1 P00915 1/20 0.53
CA2 P00918 1/20 0.53
MTNR1A P48039 2/20 0.52
MTNR1B P49286 2/20 0.52
IDO1 P14902 1/20 0.49
RAB9A P51151 1/20 0.49
POLB P06746 1/20 0.47
CNR1 P21554 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5195352 0.86 ALDH1A1 (0.58) KDM4EALDH1A1CA1CA2POLB
SCHEMBL11475368 0.84 EPHX2 (0.67) KDM4EALDH1A1CA1CA2MTNR1A
SCHEMBL5191195 0.83 MEN1 (0.59) KDM4EALDH1A1CA1CA2
SCHEMBL5213635 0.79 KDM4E (0.53) KDM4EALDH1A1CA1CA2MTNR1A
SCHEMBL11654998 0.78 CA1 (0.77) ALDH1A1CA1CA2MTNR1AMTNR1B
SCHEMBL5195710 0.78 ALDH1A1 (0.58) ALDH1A1CA1CA2RAB9APOLB
SCHEMBL29557686 0.77 POLB (0.60) ALDH1A1POLB
SCHEMBL3347513 0.77 POLB (0.60) ALDH1A1POLB
Hydrochloric Acid SCHEMBL11659562 0.77 CA1 (0.76) ALDH1A1CA1CA2MTNR1AMTNR1B
SCHEMBL30475090 0.76 POLB (0.59) ALDH1A1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0968206-B8 N-HETEROCYCLIC DERIVATIVES AS NOS INHIBITORS BERLEX INC (US) 2007-01-24 EP claimed
EP-0968206-A1 N-HETEROCYCLIC DERIVATIVES AS NOS INHIBITORS BERLEX LABORATORIES, INC. (US) 2000-01-05 EP claimed
WO-1998037079-A1 N-HETEROCYCLIC DERIVATIVES AS NOS INHIBITORS BERLEX LABORATORIES, INC. (US) 1998-08-27 WO claimed