SCHEMBL5218332

SCHEMBL5218332

CS(=O)(=O)c1ccc([C@@H](CCN2CCC(CCc3cc([N+](=O)[O-])ccc3S(N)(=O)=O)CC2)c2cc(F)cc(F)c2)cc1

nearest known ligand 0.49

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 19/20 0.49
KCNH2 Q12809 2/20 0.49
CYP2D6 P10635 1/20 0.49
KCNJ1 P48048 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5218232 0.82 CCR5 (0.53) CCR5KCNH2CYP2D6KCNJ1
SCHEMBL5219971 0.80 CCR5 (0.60) CCR5KCNH2CYP2D6
SCHEMBL5222946 0.80 CCR5 (0.54) CCR5KCNH2CYP2D6KCNJ1
SCHEMBL5220283 0.78 CCR5 (0.61) CCR5KCNH2CYP2D6
SCHEMBL3303563 0.78 CCR5 (0.59) CCR5KCNH2CYP2D6
Hydrochloric Acid SCHEMBL5222702 0.78 CCR5 (0.61) CCR5KCNH2CYP2D6
SCHEMBL5238997 0.77 CCR5 (0.58) CCR5KCNH2CYP2D6
SCHEMBL5235987 0.77 CCR5 (0.61) CCR5KCNH2CYP2D6
SCHEMBL5220551 0.76 CCR5 (0.61) CCR5KCNH2CYP2D6
SCHEMBL5434212 0.74 CCR5 (0.62) CCR5KCNH2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1654229-B1 PIPERIDINE DERIVATIVES AS CCR5 RECEPTOR MODULATORS ASTRAZENECA AB (SE) 2007-05-09 EP disclosed