SCHEMBL5219741

SCHEMBL5219741

C[C@@H](c1ccccc1)n1c(CN2CCOCC2)nnc1CN1CCN(c2ccccn2)CC1

nearest known ligand 0.56

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
AVPR1A P37288 2/20 0.56
GRM2 Q14416 1/20 0.47
HTR1A P08908 1/20 0.47
KDM4E B2RXH2 4/20 0.45
ALDH1A1 P00352 4/20 0.45
TDP1 Q9NUW8 1/20 0.45
KCNH2 Q12809 1/20 0.45
HPGD P15428 1/20 0.45
HSD17B10 Q99714 1/20 0.45
MAPT P10636 2/20 0.44
LMNA P02545 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
DRD4 P21917 1/20 0.43
NPC1 O15118 1/20 0.43
HTT P42858 1/20 0.43
RAB9A P51151 1/20 0.43
SLC6A2 P23975 2/20 0.43
SLC6A3 Q01959 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL5211533 0.99 AVPR1A (0.55) AVPR1AGRM2HTR1AKDM4EALDH1A1
Hydrochloric Acid SCHEMBL5211525 0.99 AVPR1A (0.55) AVPR1AGRM2HTR1AKDM4EALDH1A1
SCHEMBL5212007 0.90 ALDH1A1 (0.48) AVPR1AHTR1AKDM4EALDH1A1MAPT
Hydrochloric Acid SCHEMBL5211566 0.89 ALDH1A1 (0.47) AVPR1AHTR1AKDM4EALDH1A1MAPT
Hydrochloric Acid SCHEMBL5211577 0.89 ALDH1A1 (0.47) AVPR1AHTR1AKDM4EALDH1A1MAPT
SCHEMBL5215865 0.77 AVPR1A (0.59) AVPR1A
SCHEMBL11059996 0.76 KCNH2 (0.67) HTR1AKDM4EALDH1A1TDP1KCNH2
SCHEMBL5215034 0.76 MAPT (0.64) AVPR1AKDM4EALDH1A1TDP1KCNH2
SCHEMBL5215652 0.74 AVPR1A (0.55) AVPR1A
SCHEMBL11062709 0.72 ALDH1A1 (0.52) KDM4EALDH1A1KCNH2HPGDHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1558598-B1 TRIAZOLE COMPOUNDS FOR THE TREATMENT OF DYSMENORRHOEA PFIZER LTD (GB) 2007-07-18 EP claimed