SCHEMBL5219926

SCHEMBL5219926

C1=CC2(c3ccc(-c4cccc5cccnc45)nc3)CCN(C1)C2

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 1/20 0.36
CCNC P24863 1/20 0.32
CDK8 P49336 1/20 0.32
HTR2A P28223 3/20 0.31
HTR2C P28335 3/20 0.31
HTR2B P41595 2/20 0.31
KDM4E B2RXH2 1/20 0.31
GMNN O75496 1/20 0.31
LMNA P02545 1/20 0.31
TP53 P04637 1/20 0.31
HSP90AA1 P07900 1/20 0.31
MMP2 P08253 1/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2D6 P10635 1/20 0.31
MAPT P10636 1/20 0.31
MMP9 P14780 1/20 0.31
ALOX15 P16050 1/20 0.31
TSHR P16473 1/20 0.31
NFKB1 P19838 1/20 0.31
MMP8 P22894 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bromide SCHEMBL4558860 0.99 CNR2 (0.36) CNR2CCNCCDK8HTR2AHTR2C
SCHEMBL2677975 0.83 CNR2 (0.41) CNR2CCNCCDK8HTR2AHTR2C
SCHEMBL4465415 0.81 NPC1 (0.36)
SCHEMBL5220383 0.79 CNR2 (0.38) CNR2CCNCCDK8HTR2AHTR2C
Bromide SCHEMBL4558553 0.78 CNR2 (0.38) CNR2CCNCCDK8HTR2AHTR2C
SCHEMBL5219426 0.78 HSD11B1 (0.32)
SCHEMBL4483243 0.78 CYP2A6 (0.41) KDM4EHSP90AA1CYP3A4CYP2D6TSHR
Bromide SCHEMBL4460345 0.77 HSD11B1 (0.31)
SCHEMBL4463819 0.77 HSD11B1 (0.38)
SCHEMBL4463770 0.76 ALOX5AP (0.34) ALOX5AP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1465893-B1 DERIVATIVES OF 5-(PYRIDIN-3-YL)-1-AZABICYCLO (3.2.1) OCTANE, THE PREPARATION THEREOF AND THE APPLICATION OF SAME IN THERAPEUTICS SANOFI AVENTIS (FR) 2007-02-28 EP claimed