SCHEMBL5220871

SCHEMBL5220871

COC(=N)Cc1c(Cl)cccc1Cl

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1B1 P15121 1/20 0.48
KMT2A Q03164 3/20 0.43
SMN1; SMN2 Q16637 4/20 0.42
ADRA2A P08913 2/20 0.41
CYP3A4 P08684 2/20 0.41
CYP2C9 P11712 2/20 0.41
MAPK1 P28482 2/20 0.41
CYP2C19 P33261 2/20 0.41
MEN1 O00255 1/20 0.41
LMNA P02545 1/20 0.41
HTR1A P08908 1/20 0.41
CYP2D6 P10635 1/20 0.41
ADRA2B P18089 1/20 0.41
ADRA2C P18825 1/20 0.41
MAOA P21397 1/20 0.41
ADRA1D P25100 1/20 0.41
HTR2A P28223 1/20 0.41
HTR2C P28335 1/20 0.41
ADRA1A P35348 1/20 0.41
DRD3 P35462 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL5219918 0.98 AKR1B1 (0.47) AKR1B1KMT2ASMN1; SMN2ADRA2ACYP3A4
SCHEMBL3743731 0.76 AKR1B1 (0.59) AKR1B1KMT2ASMN1; SMN2ADRA2ACYP3A4
SCHEMBL14464764 0.74 AKR1B1 (0.56) AKR1B1KMT2ASMN1; SMN2ADRA2ACYP3A4
SCHEMBL837827 0.73 AKR1B1 (0.50) AKR1B1KMT2ASMN1; SMN2ADRA2ACYP3A4
SCHEMBL7637016 0.73 AKR1B1 (0.55) AKR1B1KMT2ASMN1; SMN2ADRA2ACYP3A4
SCHEMBL1021475 0.72 AKR1B1 (0.54) AKR1B1KMT2ASMN1; SMN2ADRA2ACYP3A4
Hydrochloric Acid SCHEMBL1182809 0.71 ADRA2A (0.55) AKR1B1KMT2ASMN1; SMN2ADRA2ACYP3A4
SCHEMBL23102301 0.70 AKR1B1 (0.42) AKR1B1KMT2ASMN1; SMN2ADRA2ACYP3A4
Hydrochloric Acid SCHEMBL29195762 0.70 KMT2A (0.51) KMT2ASMN1; SMN2MEN1LMNAMAPT
SCHEMBL10308335 0.68 AKR1B1 (0.41) AKR1B1KMT2ASMN1; SMN2ADRA2ACYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7265138-B2 Vanilloid receptor ligands and their use in treatments AMGEN INC. (US) 2007-09-04 US disclosed
US-7265138-B2 Vanilloid receptor ligands and their use in treatments AMGEN INC. (US) 2007-09-04 US disclosed
EP-1818333-A1 Vanilloid receptor ligands and their use in treatments Amgen Inc. (US) 2007-08-15 EP disclosed
EP-1818333-A1 Vanilloid receptor ligands and their use in treatments Amgen Inc. (US) 2007-08-15 EP disclosed