SCHEMBL5221354

SCHEMBL5221354

CCC(CC)Nc1nc(Cl)nc2c1ncn2C1OC(c2nnn(CC)n2)C(O)C1O

nearest known ligand 0.81

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 19/20 0.81
ADORA2A P29274 19/20 0.81
ADORA1 P30542 19/20 0.81
ADORA2B P29275 15/20 0.81

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4232897 1.00 ADORA3 (0.81) ADORA3ADORA2AADORA1ADORA2B
SCHEMBL10156540 0.89 ADORA3 (0.85) ADORA3ADORA2AADORA1ADORA2B
SCHEMBL11968432 0.88 ADORA3 (0.74) ADORA3ADORA2AADORA1ADORA2B
SCHEMBL2811320 0.88 ADORA3 (0.74) ADORA3ADORA2AADORA1ADORA2B
SCHEMBL3904472 0.88 ADORA3 (0.74) ADORA3ADORA2AADORA1ADORA2B
SCHEMBL10156565 0.87 ADORA3 (0.80) ADORA3ADORA2AADORA1ADORA2B
SCHEMBL10156530 0.87 ADORA3 (0.82) ADORA3ADORA2AADORA1ADORA2B
SCHEMBL10156549 0.87 ADORA3 (0.82) ADORA3ADORA2AADORA1ADORA2B
SCHEMBL3294999 0.86 ADORA3 (1.00) ADORA3ADORA2AADORA1ADORA2B
SCHEMBL10156554 0.86 ADORA3 (0.80) ADORA3ADORA2AADORA1ADORA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1861412-A1 ADENOSINE DERIVATIVES HAVING A2A RECEPTOR ACTIVITY Novartis AG (CH) 2007-12-05 EP disclosed
WO-2006097260-A1 ADENOSINE DERIVATIVES HAVING A2A RECEPTOR ACTIVITY NOVARTIS AG (CH) 2006-09-21 WO disclosed