SCHEMBL5221843

SCHEMBL5221843

Nc1ncc(-c2ccc(S(=O)(=O)N3CCCC3)cc2)nc1C(=O)NCCN1CCOCC1

nearest known ligand 0.65

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 12/20 0.65
CCNE2 O96020 9/20 0.65
CCNE1 P24864 9/20 0.65
CDK2 P24941 9/20 0.65
ATR Q13535 3/20 0.56
KCNH2 Q12809 1/20 0.55
POLB P06746 1/20 0.53
SMN1; SMN2 Q16637 1/20 0.53
GSK3A P49840 1/20 0.52
ACVR1 Q04771 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL3279262 0.99 GSK3B (0.64) GSK3BCCNE2CCNE1CDK2ATR
SCHEMBL3279536 0.95 GSK3B (0.67) GSK3BCCNE2CCNE1CDK2ATR
Hydrochloric Acid SCHEMBL6206046 0.92 GSK3B (0.59) GSK3BCCNE2CCNE1CDK2ATR
SCHEMBL3274547 0.85 GSK3B (0.78) GSK3BCCNE2CCNE1CDK2ATR
Hydrochloric Acid SCHEMBL5224249 0.85 GSK3B (0.49) GSK3BCCNE2CCNE1CDK2ATR
SCHEMBL3273882 0.84 GSK3B (0.67) GSK3BCCNE2CCNE1CDK2ATR
Hydrochloric Acid SCHEMBL4505372 0.84 CCNE2 (0.53) GSK3BCCNE2CCNE1CDK2ATR
SCHEMBL3274403 0.83 GSK3B (0.65) GSK3BCCNE2CCNE1CDK2ATR
SCHEMBL5218515 0.81 GSK3B (0.63) GSK3BCCNE2CCNE1CDK2ATR
SCHEMBL5219446 0.81 GSK3B (0.51) GSK3BCCNE2CCNE1CDK2KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1575942-B1 COMPOUNDS HAVING SELECTIVE INHIBITING EFECT AT GSK3 ASTRAZENECA AB (SE) 2007-05-02 EP claimed