SCHEMBL5221955

SCHEMBL5221955

N[C@@H](Cc1ccccc1)[C@H](O)CNCCc1cccc(C(F)(F)F)c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 4/20 0.49
BCHE P06276 3/20 0.49
HTR2A P28223 2/20 0.47
HTR2C P28335 2/20 0.47
HTR2B P41595 2/20 0.47
KDM4E B2RXH2 2/20 0.46
MEN1 O00255 1/20 0.46
KMT2A Q03164 1/20 0.46
TAAR1 Q96RJ0 1/20 0.46
CYP3A4 P08684 3/20 0.46
CYP1A2 P05177 2/20 0.46
CYP2D6 P10635 2/20 0.46
TP53 P04637 1/20 0.46
TSHR P16473 1/20 0.46
CYP2C19 P33261 1/20 0.46
SIGMAR1 Q99720 1/20 0.46
TDP1 Q9NUW8 1/20 0.44
USP2 O75604 2/20 0.43
NR1I2 O75469 1/20 0.43
ADRB1 P08588 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL161260 0.88 BACE1 (0.62) BACE1BCHEHTR2AHTR2CHTR2B
SCHEMBL3455222 0.88 BACE1 (0.62) BACE1BCHEHTR2AHTR2CHTR2B
SCHEMBL8276492 0.88 BACE1 (0.62) BACE1BCHEHTR2AHTR2CHTR2B
Hydrochloric Acid SCHEMBL2499284 0.87 BACE1 (0.61) BACE1BCHEHTR2AHTR2CHTR2B
SCHEMBL3354800 0.84 TAAR1 (0.46) KDM4ETAAR1OPRM1
Formic Acid SCHEMBL5928562 0.84 BACE1 (0.60) BACE1BCHEHTR2AHTR2CHTR2B
SCHEMBL4044665 0.83 ANPEP (0.55) BCHECYP3A4CYP1A2CYP2D6TSHR
SCHEMBL496056 0.83 ANPEP (0.55) BCHECYP3A4CYP1A2CYP2D6TSHR
SCHEMBL3347864 0.83 ANPEP (0.55) BCHECYP3A4CYP1A2CYP2D6TSHR
SCHEMBL4696783 0.83 ANPEP (0.55) BCHECYP3A4CYP1A2CYP2D6TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1567488-B1 HYDROXYETHYLAMINE DERIVATIVES FOR THE TREATMENT OF ALZHEIMER'S DISEASE GLAXO GROUP LTD (GB) 2007-02-21 EP disclosed