SCHEMBL5222045

SCHEMBL5222045

COc1ccc(CC(O)CN2C[CH]N(C3CCCCC3)CC2)cc1

nearest known ligand 0.54

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 1/20 0.54
KDM4E B2RXH2 1/20 0.44
POLB P06746 1/20 0.44
KMT2A Q03164 3/20 0.41
ALDH1A1 P00352 1/20 0.41
TSHR P16473 1/20 0.41
LMNA P02545 1/20 0.40
MAPK1 P28482 1/20 0.40
HTT P42858 1/20 0.40
MEN1 O00255 2/20 0.40
DRD4 P21917 1/20 0.40
SLC18A2 Q05940 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6256736 0.99 CYP2D6 (0.55) CYP2D6KDM4EPOLBKMT2AALDH1A1
SCHEMBL6256508 0.89 KMT2A (0.44) CYP2D6KDM4EPOLBKMT2AALDH1A1
SCHEMBL6259368 0.88 SLC18A2 (0.43) CYP2D6KDM4EPOLBKMT2AALDH1A1
SCHEMBL6188797 0.74 CYP2D6 (0.55) CYP2D6KDM4EPOLBKMT2AALDH1A1
SCHEMBL7705235 0.73 CYP2D6 (0.54) CYP2D6KMT2ALMNAMAPK1HTT
SCHEMBL4500156 0.73 EPHX2 (0.59) CYP2D6KDM4EPOLBALDH1A1TSHR
SCHEMBL4503243 0.72 EPHX2 (0.57) CYP2D6KDM4EKMT2ALMNADRD4
SCHEMBL5226751 0.71 CYP2D6 (0.54) CYP2D6LMNAMAPK1HTT
SCHEMBL8734239 0.70 SLC18A3 (0.72) CYP2D6ALDH1A1LMNADRD4
SCHEMBL6256607 0.68 CYP2D6 (0.47) CYP2D6KMT2ALMNAMAPK1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1806346-A1 Substituted piperazine compounds and their use as fatty acid oxidation inhibitors CV THERAPEUTICS, INC. (US) 2007-07-11 EP disclosed
EP-1578737-A1 SUBSTITUTED HETEROCYCLIC COMPOUNDS CV THERAPEUTICS, INC. (US) 2005-09-28 EP disclosed
EP-1567525-A2 SUBSTITUTED PIPERAZINE COMPOUNDS AND THEIR USE AS FATTY ACID OXIDATION INHIBITORS CV THERAPEUTICS, INC. (US) 2005-08-31 EP disclosed
WO-2004063180-A1 SUBSTITUTED HETEROCYCLIC COMPOUNDS CV THERAPEUTICS, INC. (US) 2004-07-29 WO disclosed
WO-2004052887-A2 SUBSTITUTED PIPERAZINE COMPOUNDS AND THEIR USE AS FATTY ACID OXIDATION INHIBITORS CV THERAPEUTICS, INC. (US) 2004-06-24 WO disclosed