SCHEMBL5222419

SCHEMBL5222419

CCc1nc2cc(OCC(O)CN3C[CH]N(c4nc5ccccc5s4)CC3)ccc2s1

nearest known ligand 0.48

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.45
CYP1A2 P05177 2/20 0.45
CYP2C9 P11712 2/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6184015 0.90 CYP3A4 (0.56) CYP3A4CYP1A2CYP2C9
SCHEMBL6205691 0.80 KCNH2 (0.51) CYP3A4CYP1A2CYP2C9
SCHEMBL5224373 0.80 IDO1 (0.48) CYP3A4CYP1A2CYP2C9
SCHEMBL4862557 0.78 CYP3A4 (0.63) CYP3A4CYP1A2CYP2C9
SCHEMBL4036205 0.78 CYP3A4 (0.50) CYP3A4CYP1A2CYP2C9
SCHEMBL6259496 0.75 RAB9A (0.54) CYP1A2CYP2C9
SCHEMBL7005719 0.74 CYP3A4 (0.52) CYP3A4CYP1A2CYP2C9
SCHEMBL4867229 0.74 CYP3A4 (0.61) CYP3A4CYP1A2CYP2C9
SCHEMBL4035200 0.74 CYP3A4 (0.61) CYP3A4CYP1A2CYP2C9
SCHEMBL5965204 0.73 CYP3A4 (0.52) CYP3A4CYP1A2CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1806346-A1 Substituted piperazine compounds and their use as fatty acid oxidation inhibitors CV THERAPEUTICS, INC. (US) 2007-07-11 EP disclosed
EP-1567525-A2 SUBSTITUTED PIPERAZINE COMPOUNDS AND THEIR USE AS FATTY ACID OXIDATION INHIBITORS CV THERAPEUTICS, INC. (US) 2005-08-31 EP disclosed
WO-2004052887-A2 SUBSTITUTED PIPERAZINE COMPOUNDS AND THEIR USE AS FATTY ACID OXIDATION INHIBITORS CV THERAPEUTICS, INC. (US) 2004-06-24 WO disclosed