SCHEMBL5222857

SCHEMBL5222857

CC(Oc1ccc(S(C)(=O)=O)cc1C(=O)N1Cc2cc(C(F)(F)F)cnc2C1)C(F)(F)F

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
SLC6A9 P48067 20/20 1.00
SLC6A5 Q9Y345 3/20 0.68
KCNH2 Q12809 3/20 0.67

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1461318 1.00 SLC6A9 (1.00) SLC6A9SLC6A5KCNH2
SCHEMBL3871601 1.00 SLC6A9 (1.00) SLC6A9SLC6A5KCNH2
SCHEMBL18490920 0.94 SLC6A9 (0.89) SLC6A9SLC6A5KCNH2
SCHEMBL3872054 0.93 SLC6A9 (1.00) SLC6A9SLC6A5KCNH2
SCHEMBL3878358 0.91 SLC6A9 (0.84) SLC6A9SLC6A5KCNH2
SCHEMBL18502987 0.90 SLC6A9 (0.82) SLC6A9SLC6A5
SCHEMBL9882712 0.90 SLC6A9 (0.84) SLC6A9SLC6A5KCNH2
SCHEMBL9882711 0.90 SLC6A9 (0.84) SLC6A9SLC6A5KCNH2
SCHEMBL3871584 0.90 SLC6A9 (0.81) SLC6A9SLC6A5
SCHEMBL3880029 0.89 SLC6A9 (0.80) SLC6A9SLC6A5KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106163520-B GLYT1 inhibitors for the treatment of hematological disorders 豪夫迈·罗氏有限公司 2019-12-13 CN claimed
CN-106163520-B GLYT1 inhibitors for the treatment of hematological disorders 豪夫迈·罗氏有限公司 2019-12-13 CN disclosed
EP-3137073-B1 GLYT1 INHIBITORS FOR USE IN THE TREATMENT OF HEMATOLOGICAL DISORDERS HOFFMANN LA ROCHE (CH) 2018-06-06 EP disclosed
EP-1848694-A1 HETEROCYCLIC SUBSTITUTED PHENYL METHANONES AS INHIBITORS OF THE GLYCINE TRANSPORTER 1 F. Hoffmann-Roche AG (CH) 2007-10-31 EP disclosed
WO-2006082001-A1 HETEROCYCLIC SUBSTITUTED PHENYL METHANONES AS INHIBITORS OF THE GLYCINE TRANSPORTER 1 F.HOFFMANN-LA ROCHE AG (CH) 2006-08-10 WO disclosed