SCHEMBL5223011

SCHEMBL5223011

COc1ccc(-c2ccc(C34CCCN(CC3)C4)cn2)cc1OC

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FYN P06241 5/20 0.40
ALDH1A1 P00352 4/20 0.39
KDM4E B2RXH2 3/20 0.39
HPGD P15428 3/20 0.39
HSD17B10 Q99714 2/20 0.39
MAPK1 P28482 2/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
TSHR P16473 1/20 0.39
CASP1 P29466 1/20 0.39
CASP7 P55210 1/20 0.39
NOS1 P29475 1/20 0.38
SLC6A2 P23975 1/20 0.37
SLC6A4 P31645 1/20 0.37
SLC6A3 Q01959 1/20 0.37
USP2 O75604 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2C9 P11712 1/20 0.36
ALOX15 P16050 1/20 0.36
CYP2C19 P33261 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bromide SCHEMBL4460701 0.99 FYN (0.40) FYNALDH1A1KDM4EHPGDHSD17B10
SCHEMBL2678759 0.98 FYN (0.42) FYNALDH1A1KDM4EHPGDHSD17B10
Hydrochloric Acid SCHEMBL2678564 0.97 FYN (0.41) FYNALDH1A1KDM4EHPGDHSD17B10
SCHEMBL2678945 0.95 FYN (0.43) FYNALDH1A1KDM4EHPGDHSD17B10
SCHEMBL2679330 0.88 HSD11B1 (0.41) ALDH1A1KDM4EHPGDSMN1; SMN2CYP3A4
SCHEMBL2678054 0.85 HSD11B1 (0.42) ALDH1A1KDM4EHPGDHSD17B10SMN1; SMN2
SCHEMBL4469713 0.85 RXFP1 (0.41) FYNSMN1; SMN2SLC6A2SLC6A4SLC6A3
Bromide SCHEMBL4480044 0.84 RXFP1 (0.40) FYNSMN1; SMN2SLC6A2SLC6A4SLC6A3
SCHEMBL2678305 0.83 KDM1A (0.47) FYNALDH1A1KDM4EHSD17B10SMN1; SMN2
SCHEMBL2678397 0.82 RXFP1 (0.43) FYNSMN1; SMN2NOS1SLC6A2SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1465893-B1 DERIVATIVES OF 5-(PYRIDIN-3-YL)-1-AZABICYCLO (3.2.1) OCTANE, THE PREPARATION THEREOF AND THE APPLICATION OF SAME IN THERAPEUTICS SANOFI AVENTIS (FR) 2007-02-28 EP claimed