SCHEMBL522352

SCHEMBL522352

COC(=O)/C=C/C1=CC=C(Br)CC1=S

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.38
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
TYR P14679 1/20 0.38
CA7 P43166 1/20 0.38
CA9 Q16790 1/20 0.38
CA14 Q9ULX7 1/20 0.38
TTR P02766 1/20 0.36
APP P05067 1/20 0.36
HCAR2 Q8TDS4 2/20 0.35
KEAP1 Q14145 1/20 0.35
NFE2L2 Q16236 1/20 0.35
ALDH1A1 P00352 5/20 0.35
KDM4E B2RXH2 5/20 0.35
MAPT P10636 4/20 0.35
KMT2A Q03164 3/20 0.35
MEN1 O00255 2/20 0.35
TP53 P04637 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP2C9 P11712 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL521742 0.75 CA12 (0.40) CA12CA1CA2TYRCA7
SCHEMBL29536245 0.63 HCAR2 (0.52) CA12CA1CA2TYRCA7
SCHEMBL15150027 0.61 CA12 (0.46) CA12CA1CA2CA7CA9
SCHEMBL403042 0.61 CA12 (0.70) CA12CA1CA2TYRCA7
SCHEMBL403043 0.61 CA12 (0.70) CA12CA1CA2TYRCA7
SCHEMBL5259514 0.61 CA12 (0.70) CA12CA1CA2TYRCA7
SCHEMBL6821064 0.61 AKR1C3 (0.56) CA12CA1CA2TYRCA7
SCHEMBL6821063 0.61 AKR1C3 (0.56) CA12CA1CA2TYRCA7
SCHEMBL71224 0.61 CA12 (0.84) CA12CA1CA2TYRCA7
SCHEMBL5057418 0.61 CA12 (0.84) CA12CA1CA2TYRCA7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2417082-B1 CATALYTIC WITTIG AND MITSUNOBU REACTIONS UNIV TEXAS (US) 2016-03-16 EP disclosed
US-8901365-B2 Catalytic Wittig and Mitsunobu reactions BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM (US) 2014-12-02 US disclosed
EP-2417082-A2 CATALYTIC WITTIG AND MITSUNOBU REACTIONS THE BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM (US) 2012-02-15 EP disclosed
US-20120029211-A1 Catalytic Wittig and Mitsunobu Reactions THE UNIVERSITY OF TEXAS AT ARLINGTON 2012-02-02 US disclosed
WO-2010118042-A2 CATALYTIC WITTIG AND MITSUNOBU REACTIONS BOARD OF REGENTS THE UNIVERSITY OF TEXAS AT ARLINGTON (US) 2010-10-14 WO disclosed